SCHEMBL22184887

SCHEMBL22184887

COc1cc(Cl)cc2cc(C(C)C)c(=O)[nH]c12

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 12/20 0.45
TRPV1 Q8NER1 2/20 0.38
PDE3B Q13370 3/20 0.38
PDE3A Q14432 3/20 0.38
ERN1 O75460 1/20 0.36
LPAR1 Q92633 1/20 0.35
GRIN2D O15399 1/20 0.35
GRIN3B O60391 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2A Q12879 1/20 0.35
GRIN2B Q13224 1/20 0.35
GRIN2C Q14957 1/20 0.35
GRIN3A Q8TCU5 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22184888 0.83 IDH1 (0.36) IDH1TRPV1
SCHEMBL22185210 0.81 PDE3B (0.40) IDH1TRPV1PDE3BPDE3A
SCHEMBL22198974 0.80 IDH1 (0.47) IDH1PDE3BPDE3AERN1GRIN2D
SCHEMBL21549766 0.79 IDH1 (0.49) IDH1TRPV1GRIN2DGRIN3BGRIN1
SCHEMBL17603389 0.78 IDH1 (0.55) IDH1
SCHEMBL17603348 0.78 ERN1 (0.50) IDH1PDE3BPDE3AERN1GRIN2D
SCHEMBL22185229 0.78 IDH1 (0.57) IDH1PDE3BPDE3A
SCHEMBL22185212 0.77 CNR2 (0.48) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL22184879 0.75 EIF4A3 (0.45) TRPV1PDE3BPDE3AGRIN2DGRIN3B
SCHEMBL20559286 0.75 CNR2 (0.53) IDH1ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200206233-A1 HETEROCYCLIC COMPOUNDS AS MUTANT IDH INHIBITORS INTEGRAL BIOSCIENCES PRIVATE LIMITED (IN) 2020-07-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200206233-A1 HETEROCYCLIC COMPOUNDS AS MUTANT IDH INHIBITORS IDH1, IDH2, IDH3A IDH1 1/4885TRPV1 4635/4885PDE3B 1672/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.