SCHEMBL22199033

SCHEMBL22199033

Cc1cn(-c2ccc(OC(F)(F)F)c(F)c2)cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR2E1 Q9Y466 3/20 0.44
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP19A1 P11511 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
MAOA P21397 3/20 0.42
MAOB P27338 3/20 0.42
PSEN1 P49768 3/20 0.41
PSEN2 P49810 3/20 0.41
APH1B Q8WW43 3/20 0.41
NCSTN Q92542 3/20 0.41
APH1A Q96BI3 3/20 0.41
PSENEN Q9NZ42 3/20 0.41
USP30 Q70CQ3 2/20 0.40
CYP2E1 P05181 1/20 0.39
CYP2A6 P11509 1/20 0.39
PDE2A O00408 1/20 0.38
EPHX2 P34913 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22199042 0.87 NR2E1 (0.45) NR2E1CYP1A2CYP3A4CYP2D6CYP19A1
SCHEMBL22199043 0.84 MAOA (0.53) NR2E1CYP1A2CYP3A4CYP2D6CYP19A1
SCHEMBL22185266 0.83 PDE2A (0.38) NR2E1PDE2AEPHX2
SCHEMBL22185883 0.83 PDE2A (0.39) PDE2AEPHX2
SCHEMBL22199017 0.78 CYP1A2 (0.59) NR2E1CYP1A2CYP3A4CYP2D6CYP19A1
SCHEMBL22184923 0.77 KCNH2 (0.48) NR2E1CYP1A2CYP3A4CYP2D6CYP19A1
SCHEMBL971611 0.77 MAPT (0.39) NR2E1CYP1A2CYP3A4CYP2D6CYP19A1
SCHEMBL22198918 0.74 CYP1A2 (0.46) NR2E1CYP1A2CYP3A4CYP2D6CYP19A1
SCHEMBL22185264 0.74 SCN5A (0.40) NR2E1MAOAMAOBGRM2
SCHEMBL7921146 0.73 PSEN1 (0.48) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020141439-A1 HETEROCYCLIC COMPOUNDS AS MUTANT IDH INHIBITORS INTEGRAL BIOSCIENCES PRIVATE LIMITED (IN) 2020-07-09 WO disclosed