SCHEMBL22200575

SCHEMBL22200575

CC(C)n1c(=O)c(-c2c(F)cc(NSCc3ccc(F)cc3)c(F)c2F)cc2cnc(N)nc21

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 2/20 0.43
BRAF P15056 2/20 0.42
BTK Q06187 1/20 0.39
EGFR P00533 1/20 0.36
FGFR1 P11362 1/20 0.36
SRC P12931 1/20 0.36
FGFR2 P21802 1/20 0.36
FGFR4 P22455 1/20 0.36
FGFR3 P22607 1/20 0.36
ABL1 P00519 1/20 0.34
PIK3CA P42336 2/20 0.34
MTOR P42345 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22200771 0.89 ERN1 (0.40) ERN1BRAFBTKEGFRFGFR1
SCHEMBL22200577 0.89 ERN1 (0.49) ERN1BRAFBTKEGFRFGFR1
SCHEMBL22200366 0.86 ERN1 (0.47) ERN1BRAFBTKEGFRFGFR1
SCHEMBL25034102 0.85 ERN1 (0.55) ERN1BRAFBTKEGFRFGFR1
SCHEMBL22200568 0.84 ERN1 (0.41) ERN1BRAFBTKEGFRFGFR1
SCHEMBL22200582 0.82 PIK3CA (0.43) ERN1BRAFBTKEGFRFGFR1
SCHEMBL22200612 0.79 RORC (0.35) ERN1BRAFBTK
SCHEMBL22200701 0.78 ERN1 (0.42) ERN1BRAFBTKEGFRFGFR1
SCHEMBL22200371 0.78 PIK3CA (0.38) BRAFBTKEGFRFGFR1SRC
SCHEMBL25034168 0.77 ERN1 (0.68) ERN1BRAFBTKEGFRFGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020142612-A1 PYRIDO-PYRIMIDINONE AND PTERIDINONE COMPOUNDS AS INHIBITORS OF ENDORIBONUCLEASE INOSITOL REQUIRING ENZYME I (IRE I ALPHA) FOR THE TREATMENT OF CANCER DISEASES. GENENTECH, INC. (US) 2020-07-09 WO disclosed