SCHEMBL22201144

SCHEMBL22201144

O=C1CC[C@@H](c2ccc(C(F)(F)F)cc2)N1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.48
PARP2 Q9UGN5 1/20 0.48
DDB1 Q16531 3/20 0.48
CRBN Q96SW2 3/20 0.48
HTR2C P28335 2/20 0.46
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
CMA1 P23946 1/20 0.40
HDAC11 Q96DB2 1/20 0.39
HDAC2 Q92769 1/20 0.39
KIF11 P52732 1/20 0.39
TACR1 P25103 1/20 0.39
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
ESR1 P03372 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22190351 1.00 PARP1 (0.48) PARP1PARP2DDB1CRBNHTR2C
SCHEMBL8530446 0.90 PARP1 (0.46) PARP1PARP2DDB1CRBNHTR2C
SCHEMBL22201150 0.83 DDB1 (0.47) DDB1CRBNPDE4APDE4BPDE4C
SCHEMBL14457994 0.83 DDB1 (0.47) DDB1CRBNPDE4APDE4BPDE4C
SCHEMBL3600762 0.81 HTR2C (0.51) HTR2CPDE4APDE4BPDE4CPDE4D
SCHEMBL30640419 0.81 HTR2C (0.51) HTR2CPDE4APDE4BPDE4CPDE4D
SCHEMBL3600768 0.81 HTR2C (0.51) HTR2CPDE4APDE4BPDE4CPDE4D
SCHEMBL23878342 0.80 TDP1 (0.46) DDB1CRBNPDE4APDE4BPDE4C
SCHEMBL22039449 0.80 TDP1 (0.46) DDB1CRBNPDE4APDE4BPDE4C
SCHEMBL7237762 0.80 TDP1 (0.46) DDB1CRBNPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020141734-A1 METHOD FOR PREPARING CHIRAL GAMMA-LACTAM COMPOUND AND METAL COMPLEX THEREFOR 기초과학연구원 2020-07-09 WO disclosed