SCHEMBL22202070

SCHEMBL22202070

O=C1Cc2cc(-c3cncnc3)ccc2N1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.71
PDE3A Q14432 2/20 0.71
CYP11B1 P15538 4/20 0.71
CYP11B2 P19099 4/20 0.71
CYP1A2 P05177 3/20 0.71
PGR P06401 3/20 0.57
BMPR1B O00238 1/20 0.57
BMPR1A P36894 1/20 0.57
TGFBR1 P36897 1/20 0.57
ACVRL1 P37023 1/20 0.57
ACVR1 Q04771 1/20 0.57
GRIA1 P42261 3/20 0.54
CACNG8 Q8WXS5 2/20 0.54
CYP2C9 P11712 1/20 0.54
TBXAS1 P24557 1/20 0.54
AHR P35869 1/20 0.51
PDE4A P27815 1/20 0.50
PDE4B Q07343 1/20 0.50
PDE4C Q08493 1/20 0.50
PDE4D Q08499 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6746651 0.87 CYP11B1 (0.55) PDE3BPDE3ACYP11B1CYP11B2CYP1A2
SCHEMBL1119981 0.86 CYP11B1 (0.72) PDE3BPDE3ACYP11B1CYP11B2CYP1A2
SCHEMBL23143482 0.83 PDE3B (1.00) PDE3BPDE3ACYP11B1CYP11B2CYP1A2
SCHEMBL29899595 0.83 CYP11B1 (1.00) PDE3BPDE3ACYP11B1CYP11B2CYP1A2
SCHEMBL29849827 0.83 CYP11B1 (1.00) PDE3BPDE3ACYP11B1CYP11B2CYP1A2
SCHEMBL748904 0.83 CYP11B1 (1.00) PDE3BPDE3ACYP11B1CYP11B2CYP1A2
SCHEMBL29849907 0.83 CYP11B1 (1.00) PDE3BPDE3ACYP11B1CYP11B2CYP1A2
SCHEMBL1874478 0.82 CYP1A2 (0.64) PDE3BPDE3ACYP11B1CYP11B2CYP1A2
SCHEMBL3132725 0.80 PGR (0.73) PDE3BPDE3ACYP11B1CYP11B2CYP1A2
SCHEMBL18189648 0.79 GRIA1 (0.56) PDE3BPDE3ACYP11B1CYP11B2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020142486-A1 KINASE INHIBITOR COMPOUNDS AND COMPOSITIONS AND METHODS OF USE ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2020-07-09 WO disclosed