SCHEMBL2220774

SCHEMBL2220774

CCOc1cnc(-c2cccc(C(=O)C3=CC=CN(c4cnn(C)c4)N3)c2)nc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 2/20 0.34
KDR P35968 2/20 0.34
FGFR3 P22607 2/20 0.34
ALKBH1 Q13686 1/20 0.34
FGFR2 P21802 1/20 0.34
FGFR4 P22455 1/20 0.34
RIPK2 O43353 1/20 0.33
ALDH1A1 P00352 1/20 0.33
BRD4 O60885 1/20 0.33
CCL2 P13500 1/20 0.33
TTK P33981 1/20 0.33
MAPK8 P45983 1/20 0.33
RXRA P19793 1/20 0.33
RXRB P28702 1/20 0.33
ALK Q9UM73 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
IRAK4 Q9NWZ3 1/20 0.33
NPC1 O15118 1/20 0.33
TSHR P16473 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2264667 0.75 POLB (0.41) KDRFGFR3ALKBH1FGFR2FGFR4
SCHEMBL13274645 0.70 NPC1 (0.33) KDRFGFR3ALKBH1FGFR2FGFR4
SCHEMBL13449435 0.70 POLB (0.40) KDRFGFR3ALKBH1ALDH1A1RXRA
SCHEMBL2271726 0.67 ENPP2 (0.34) ENPP2IRAK4
SCHEMBL2224149 0.65 BRD4 (0.35) KDRFGFR3ALKBH1FGFR2FGFR4
SCHEMBL2221611 0.65 BRD4 (0.36) ENPP2KDRFGFR3ALKBH1BRD4
SCHEMBL13449340 0.64 BRD4 (0.34) KDRFGFR3ALKBH1BRD4CCL2
SCHEMBL164227 0.64 BRD4 (0.37) ENPP2KDRFGFR3FGFR2BRD4
SCHEMBL173429 0.64 BRD4 (0.34) ENPP2BRD4CCL2IRAK4
SCHEMBL2709532 0.64 NPC1 (0.54) RXRARXRBSMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011084402-A1 TYROSINE KINASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-07-14 WO disclosed