SCHEMBL22216321

SCHEMBL22216321

N=Cc1c(N)cc[nH]c1=O

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.43
AURKB Q96GD4 1/20 0.43
INCENP Q9NQS7 1/20 0.43
PARP1 P09874 2/20 0.41
RECQL P46063 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
JAK2 O60674 1/20 0.40
RPS6KA3 P51812 1/20 0.40
MELK Q14680 1/20 0.40
STK24 Q9Y6E0 1/20 0.40
MAPT P10636 3/20 0.36
DYRK1A Q13627 1/20 0.32
DAO P14920 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22216142 0.71 TSHR (0.33)
SCHEMBL5111881 0.70
SCHEMBL10601219 0.67
SCHEMBL10602026 0.67
SCHEMBL17005899 0.67
SCHEMBL10602635 0.67
SCHEMBL1958166 0.67
SCHEMBL18519983 0.65 KDM4E (0.41) PARP1
SCHEMBL16623599 0.65 AURKA (0.42) AURKAAURKBINCENPPARP1RECQL
SCHEMBL27314195 0.65 AURKA (0.42) AURKAAURKBINCENPPARP1RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3892621-A1 HALOALLYLAMINE COMPOUNDS AND APPLICATION THEREOF Nanjing Transthera Biosciences Co., Ltd. (CN) 2021-10-13 EP disclosed
WO-2020143763-A1 HALOALLYLAMINE COMPOUNDS AND APPLICATION THEREOF 南京药捷安康生物科技有限公司 2020-07-16 WO disclosed