SCHEMBL22220102

SCHEMBL22220102

CC(C)(C)OC(=O)N1CC2CC1CN2c1nc(Cl)nc2c(F)c(Cl)ncc12

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.45
GPR119 Q8TDV5 3/20 0.42
HDAC1 Q13547 2/20 0.41
HSD11B1 P28845 1/20 0.37
MAPK8 P45983 1/20 0.37
RET P07949 2/20 0.36
SPR P35270 1/20 0.34
PIK3CD O00329 2/20 0.34
CCR2 P41597 1/20 0.33
GRM2 Q14416 1/20 0.33
F13A1 P00488 1/20 0.33
TGM2 P21980 1/20 0.33
TGM1 P22735 1/20 0.33
KCNK3 O14649 2/20 0.33
KCNK9 Q9NPC2 2/20 0.33
SCN9A Q15858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30864079 1.00 PARP1 (0.45) PARP1GPR119HDAC1HSD11B1MAPK8
SCHEMBL25782277 1.00 PARP1 (0.45) PARP1GPR119HDAC1HSD11B1MAPK8
SCHEMBL27075129 0.93 GPR119 (0.42) PARP1GPR119HDAC1GRM2KCNK3
SCHEMBL25991254 0.88 PARP1 (0.34) PARP1GPR119HDAC1SCN9A
SCHEMBL25538247 0.85 PARP1 (0.45) PARP1GPR119HDAC1HSD11B1MAPK8
SCHEMBL24663598 0.85 SCN9A (0.38) GPR119RETPIK3CDSCN9A
SCHEMBL27003346 0.84 PARP1 (0.43) PARP1GPR119HDAC1HSD11B1MAPK8
SCHEMBL30760013 0.84 PARP1 (0.43) PARP1GPR119HDAC1HSD11B1MAPK8
SCHEMBL30966207 0.84 PARP1 (0.39) PARP1GPR119HDAC1HSD11B1MAPK8
SCHEMBL30664866 0.84 GPR119 (0.42) GPR119SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020146613-A1 KRAS G12C INHIBITORS Mirati Therapeutics, Inc. (US) 2020-07-16 WO disclosed