SCHEMBL2222993

SCHEMBL2222993

CS(=O)(=O)c1cnc(N2CCC(CC(=O)N(c3ccc(F)cc3)C3CC3)CC2)c(NC(=O)c2cccc(Cl)c2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 2/20 0.48
IDO1 P14902 3/20 0.38
SIRT2 Q8IXJ6 1/20 0.38
ATM Q13315 1/20 0.37
CCNE1 P24864 2/20 0.37
CDK2 P24941 2/20 0.37
GPR6 P46095 3/20 0.36
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
TNF P01375 1/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36
CRHBP P24387 1/20 0.36
CRHR2 Q13324 1/20 0.36
NOD2 Q9HC29 1/20 0.36
NOD1 Q9Y239 1/20 0.36
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2277699 0.88 CXCR3 (0.51) CXCR3ATMLMNASMN1; SMN2MEN1
SCHEMBL2266630 0.85 CXCR3 (0.51) CXCR3ATMLMNASMN1; SMN2HRH3
SCHEMBL2273750 0.84 CXCR3 (0.49) CXCR3IDO1GPR6LMNASMN1; SMN2
SCHEMBL12516595 0.84 CXCR3 (0.55) CXCR3ATMLMNASMN1; SMN2MEN1
SCHEMBL2271642 0.84 CXCR3 (0.49) CXCR3ATMLMNASMN1; SMN2MEN1
SCHEMBL2272027 0.84 CXCR3 (0.49) CXCR3ATMLMNASMN1; SMN2MEN1
SCHEMBL2265449 0.83 CXCR3 (0.50) CXCR3IDO1CCNE1CDK2LMNA
SCHEMBL2276798 0.82 CXCR3 (0.48) CXCR3IDO1ATMCCNE1CDK2
SCHEMBL12515556 0.82 CXCR3 (0.51) CXCR3ATMLMNASMN1; SMN2MEN1
SCHEMBL2271313 0.82 CXCR3 (0.55) CXCR3ATMLMNASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011084985-A1 CXCR3 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-07-14 WO disclosed