SCHEMBL22236258

SCHEMBL22236258

O=C(Nc1ccc(OCCN2CCCC2)nc1)c1n[nH]cc1Nc1ccc(F)c(F)c1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CD38 P28907 2/20 0.50
DYRK1A Q13627 7/20 0.48
CLK2 P49760 5/20 0.48
CLK3 P49761 3/20 0.48
MAPK1 P28482 1/20 0.45
GSK3B P49841 3/20 0.43
KDR P35968 2/20 0.42
HRH3 Q9Y5N1 1/20 0.42
KCNQ3 O43525 1/20 0.41
KCNQ2 O43526 1/20 0.41
HTR2A P28223 3/20 0.41
HTR2C P28335 3/20 0.41
WNT1 P04628 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22236260 0.90 CLK2 (0.55) CD38DYRK1ACLK2CLK3GSK3B
SCHEMBL22258274 0.82 DYRK1A (0.59) CD38DYRK1ACLK2CLK3GSK3B
SCHEMBL22236191 0.81 DYRK1A (0.55) CD38DYRK1ACLK2CLK3GSK3B
SCHEMBL22235987 0.81 DYRK1A (0.59) CD38DYRK1ACLK2CLK3GSK3B
SCHEMBL22236050 0.79 CLK2 (0.57) CD38DYRK1ACLK2CLK3HTR2A
SCHEMBL22235904 0.79 CLK2 (0.57) CD38DYRK1ACLK2CLK3GSK3B
SCHEMBL22236124 0.79 CLK2 (0.73) CD38DYRK1ACLK2CLK3GSK3B
SCHEMBL22235772 0.78 CLK2 (0.75) CD38DYRK1ACLK2CLK3GSK3B
SCHEMBL22236013 0.78 CLK2 (0.51) CD38DYRK1ACLK2CLK3GSK3B
SCHEMBL22235770 0.76 DYRK1A (0.57) CD38DYRK1ACLK2CLK3GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020150545-A1 PYRAZOLE DERIVATIVES AS MODULATORS OF THE WNT/B-CATENIN SIGNALING PATHWAY SAMUMED, LLC (US) 2020-07-23 WO disclosed