SCHEMBL22236263

SCHEMBL22236263

O=C(Nc1c[nH]nc1C(=O)Nc1ccc(C(F)(F)F)nc1)c1ccc(C(F)(F)F)nc1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 1/20 0.48
KCNH2 Q12809 1/20 0.48
TAAR1 Q96RJ0 1/20 0.48
TRPV1 Q8NER1 1/20 0.46
PTPN1 P18031 1/20 0.46
KCNQ3 O43525 3/20 0.44
KCNQ2 O43526 3/20 0.44
KCNE1 P15382 3/20 0.44
KCNQ1 P51787 3/20 0.44
CLK2 P49760 1/20 0.43
DYRK1A Q13627 1/20 0.43
CDK14 O94921 3/20 0.43
CCNY Q8ND76 3/20 0.43
P4HTM Q9NXG6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22236014 0.90 CLK2 (0.52) CLK2DYRK1A
SCHEMBL22235966 0.89 KCNQ3 (0.52) SLC6A3KCNH2TAAR1TRPV1KCNQ3
SCHEMBL22258273 0.88 KCNQ3 (0.51) TRPV1KCNQ3KCNQ2
SCHEMBL22236223 0.87 USP36 (0.50) KCNQ3KCNQ2KCNE1KCNQ1CLK2
SCHEMBL22235792 0.87 ABL1 (0.45) KCNQ3KCNQ2KCNE1KCNQ1CLK2
SCHEMBL22236228 0.87 CLK2 (0.41) TRPV1KCNQ3KCNQ2KCNE1KCNQ1
SCHEMBL22236058 0.86 USP36 (0.44) SLC6A3KCNH2TAAR1KCNQ3KCNQ2
SCHEMBL22235863 0.85 CLK2 (0.51) SLC6A3KCNH2TAAR1KCNQ3KCNQ2
SCHEMBL22236062 0.85 PTPN1 (0.42) PTPN1KCNQ3KCNQ2KCNE1KCNQ1
SCHEMBL22236081 0.81 CLK2 (0.68) CLK2DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020150545-A1 PYRAZOLE DERIVATIVES AS MODULATORS OF THE WNT/B-CATENIN SIGNALING PATHWAY SAMUMED, LLC (US) 2020-07-23 WO disclosed
WO-2020150545-A1 PYRAZOLE DERIVATIVES AS MODULATORS OF THE WNT/B-CATENIN SIGNALING PATHWAY SAMUMED, LLC (US) 2020-07-23 WO disclosed