SCHEMBL22239204

SCHEMBL22239204

COc1ccc(C(=O)CBr)nc1F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.45
KDM4E B2RXH2 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
GSK3B P49841 2/20 0.41
PTPN1 P18031 1/20 0.37
ECE1 P42892 3/20 0.37
LMNA P02545 1/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
RAB9A P51151 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
CTSA P10619 3/20 0.33
HSD11B1 P28845 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CNR2 P34972 1/20 0.33
MRGPRX4 Q96LA9 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NOD2 Q9HC29 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15595925 0.82 HPGDS (0.46) HPGDSKDM4EL3MBTL1GSK3BECE1
SCHEMBL16600772 0.76 GRIN2B (0.42) GSK3BPTPN1GRIN1GRIN2B
SCHEMBL31224297 0.75 PLK1 (0.44) HPGDSKDM4EL3MBTL1CTSACNR2
SCHEMBL16533569 0.75 CTSA (0.46) CTSA
SCHEMBL15595705 0.74 CTSA (0.56) CTSACNR2
SCHEMBL2227844 0.71 GSK3B (0.40) KDM4EL3MBTL1GSK3BPTPN1ALDH1A1
SCHEMBL24667804 0.70 CCR1 (0.42) KDM4EL3MBTL1LMNAMAPK1HTT
SCHEMBL3433496 0.70 GSK3B (0.43) HPGDSKDM4EGSK3BPTPN1CTSA
SCHEMBL31678819 0.70 GSK3B (0.43) HPGDSKDM4EGSK3BPTPN1CTSA
SCHEMBL26019074 0.70 KDM4E (0.38) KDM4EL3MBTL1LMNAHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3683207-A1 N-ALKYLARYL-5-OXYARYL-OCTAHYDRO-CYCLOPENTA[C]PYRROLE NEGATIVE ALLOSTERIC MODULATORS OF NR2B Cadent Therapeutics, Inc. (US) 2020-07-22 EP disclosed