SCHEMBL2224059

SCHEMBL2224059

Cc1cc(-c2nc3cnc(Oc4ccccc4F)nc3o2)cc(C)c1OC[C]=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.51
LMNA P02545 3/20 0.35
MAPT P10636 3/20 0.35
RXFP1 Q9HBX9 1/20 0.35
SGMS2 Q8NHU3 3/20 0.34
CEPT1 Q9Y6K0 5/20 0.33
TP53 P04637 1/20 0.33
THRB P10828 1/20 0.33
GRIN2B Q13224 1/20 0.32
DHODH Q02127 1/20 0.31
POLB P06746 1/20 0.31
PKM P14618 1/20 0.31
HTT P42858 1/20 0.31
APP P05067 1/20 0.31
USP2 O75604 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2225593 0.86 S1PR1 (0.52) S1PR1LMNAMAPTRXFP1SGMS2
SCHEMBL2225216 0.86 S1PR1 (0.69) S1PR1LMNAMAPTRXFP1CEPT1
SCHEMBL2222274 0.85 S1PR1 (0.61) S1PR1LMNAMAPTRXFP1CEPT1
SCHEMBL2222186 0.85 S1PR1 (0.48) S1PR1LMNAMAPTRXFP1SGMS2
SCHEMBL14797013 0.84 S1PR1 (0.57) S1PR1LMNAMAPTRXFP1CYP3A4
SCHEMBL2222684 0.83 S1PR1 (0.48) S1PR1LMNAMAPTRXFP1SGMS2
SCHEMBL14797187 0.81 S1PR1 (0.51) S1PR1LMNAMAPTRXFP1CEPT1
Bicarbonate SCHEMBL14486452 0.79 S1PR1 (0.50) S1PR1LMNAMAPTRXFP1CEPT1
SCHEMBL2225375 0.79 S1PR1 (0.44) S1PR1LMNAMAPTRXFP1CEPT1
SCHEMBL2228824 0.79 S1PR1 (0.42) S1PR1LMNAMAPTRXFP1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2523960-A1 HETEROCYCLIC CARBOXYLIC ACID DERIVATIVES HAVING A 2,5-SUBSTITUTED OXAZOLOPYRIMIDINE RING SANOFI (FR) 2012-11-21 EP disclosed
WO-2011086080-A1 HETEROCYCLIC CARBOXYLIC ACID DERIVATIVES HAVING A 2,5-SUBSTITUTED OXAZOLOPYRIMIDINE RING SANOFI-AVENTIS (FR) 2011-07-21 WO disclosed