SCHEMBL2224867

SCHEMBL2224867

O=C(O)c1ccccc1-c1noc(C(F)(F)F)n1

nearest known ligand 0.63

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.63
RAB9A P51151 3/20 0.63
HDAC4 P56524 12/20 0.52
HDAC6 Q9UBN7 11/20 0.50
HDAC8 Q9BY41 4/20 0.50
HDAC1 Q13547 7/20 0.48
HDAC5 Q9UQL6 3/20 0.47
HDAC3 O15379 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
KDM4E B2RXH2 1/20 0.44
USP2 O75604 1/20 0.44
ALDH1A1 P00352 1/20 0.44
TSHR P16473 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21223292 0.87 NPC1 (0.63) NPC1RAB9AHDAC4HDAC6HDAC8
SCHEMBL29975230 0.84 HDAC4 (0.55) NPC1RAB9AHDAC4HDAC6HDAC8
SCHEMBL19357146 0.83 HDAC6 (0.53) NPC1RAB9AHDAC4HDAC6HDAC8
SCHEMBL29677980 0.81 HDAC6 (0.47) NPC1RAB9AHDAC4HDAC6HDAC8
SCHEMBL30826517 0.79 HDAC6 (0.47) HDAC4HDAC6HDAC8HDAC1HDAC5
SCHEMBL27897967 0.78 CASP3 (0.62) HDAC4HDAC6HDAC8HDAC1HDAC5
SCHEMBL30102095 0.78 NPC1 (1.00) NPC1RAB9AHDAC6KDM4EALDH1A1
SCHEMBL1281643 0.77 NPC1 (0.64) NPC1RAB9AKDM4EUSP2ALDH1A1
SCHEMBL26969155 0.77 HDAC4 (0.48) HDAC4HDAC6HDAC8HDAC1HDAC5
SCHEMBL18205159 0.76 HDAC4 (0.52) HDAC4HDAC6HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112004813-B Oxadiazole compounds for controlling phytopathogenic fungi PI工业有限公司 2024-03-29 CN disclosed
CN-113788800-B Preparation method and application of 5-trifluoromethyl substituted oxadiazole compound containing diphenyl ether group 南京林业大学 2023-09-26 CN disclosed
CN-103764635-A Novel trifluoromethyl-oxadiazole derivatives and their use in the treatment of disease NOVARTIS AG 2014-04-30 CN disclosed
WO-2011088181-A9 COMPOUNDS AND METHODS TEMPERO PHARMACEUTICALS, INC. (US) 2013-01-31 WO disclosed
WO-2013006408-A1 COMPOUNDS AND METHODS TEMPERO PHARMACEUTICALS, INC. (US) 2013-01-10 WO disclosed
EP-2533783-A1 COMPOUNDS AND METHODS Tempero Pharmaceuticals, Inc. (US) 2012-12-19 EP disclosed
WO-2011088181-A1 COMPOUNDS AND METHODS TEMPERO PHARMACEUTICALS, INC. (US) 2011-07-21 WO disclosed