SCHEMBL2226690

SCHEMBL2226690

NS(=O)(=O)c1ccc(N2CCC[C@@H]2C(F)(F)F)c(CNc2cc(Nc3ccc(Cl)cc3)ncn2)c1

nearest known ligand 0.64

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TNNI3K Q59H18 17/20 0.64
CDK1 P06493 1/20 0.40
CCNB1 P14635 1/20 0.40
CCNA2 P20248 1/20 0.40
CCNE1 P24864 1/20 0.40
CDK2 P24941 1/20 0.40
CDK5 Q00535 1/20 0.40
CDK5R1 Q15078 1/20 0.40
ABL1 P00519 1/20 0.37
BCR P11274 1/20 0.37
PRCP P42785 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2225236 0.79 TNNI3K (0.51) TNNI3KCDK1CCNB1CCNA2CCNE1
SCHEMBL12517481 0.78 TNNI3K (1.00) TNNI3K
SCHEMBL14322354 0.78 TNNI3K (1.00) TNNI3K
SCHEMBL2225574 0.76 TNNI3K (0.59) TNNI3KCDK1CCNB1CCNA2CCNE1
SCHEMBL2228424 0.75 TNNI3K (0.61) TNNI3KCDK1CCNB1CCNA2CCNE1
SCHEMBL2225463 0.75 CDK1 (0.47) TNNI3KCDK1CCNB1CCNA2CCNE1
SCHEMBL2226488 0.75 TNNI3K (0.47) TNNI3KCDK1CCNB1CCNA2CCNE1
Trifluoroacetic Acid SCHEMBL14323675 0.74 TNNI3K (0.91) TNNI3K
SCHEMBL2224948 0.74 TNNI3K (0.51) TNNI3KCDK1CCNB1CCNA2CCNE1
SCHEMBL2227374 0.74 CDK1 (0.51) TNNI3KCDK1CCNB1CCNA2CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2523559-A1 COMPOUNDS AND METHODS GlaxoSmithKline LLC (US) 2012-11-21 EP claimed
WO-2011088027-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2011-07-21 WO claimed
EP-2523559-A1 COMPOUNDS AND METHODS GlaxoSmithKline LLC (US) 2012-11-21 EP disclosed
WO-2011088027-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2011-07-21 WO disclosed