SCHEMBL2226488

SCHEMBL2226488

CC1CCCN1c1ccc(S(N)(=O)=O)cc1CNc1cc(Cl)ncn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNNI3K Q59H18 5/20 0.47
SCN9A Q15858 1/20 0.37
PRCP P42785 1/20 0.35
LRRK2 Q5S007 2/20 0.35
HRH3 Q9Y5N1 3/20 0.35
KCNH2 Q12809 2/20 0.35
S1PR1 P21453 2/20 0.35
JAK3 P52333 1/20 0.34
CHRM4 P08173 1/20 0.34
WDR5 P61964 1/20 0.33
KMT2A Q03164 1/20 0.33
NPC1 O15118 1/20 0.33
HTT P42858 1/20 0.33
CDK1 P06493 1/20 0.33
CCNB1 P14635 1/20 0.33
CCNA2 P20248 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
CDK5 Q00535 1/20 0.33
CDK5R1 Q15078 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9980416 0.77 TNNI3K (0.43) TNNI3KSCN9ALRRK2HRH3KCNH2
SCHEMBL2226690 0.75 TNNI3K (0.64) TNNI3KPRCPCDK1CCNB1CCNA2
SCHEMBL2227169 0.75 CDK1 (0.40) TNNI3KCDK1CCNB1CCNA2CCNE1
SCHEMBL2227255 0.74 SLC6A4 (0.40) TNNI3KCDK1CCNB1CCNA2CCNE1
SCHEMBL14321934 0.74 TNNI3K (0.80) TNNI3KWDR5KMT2A
SCHEMBL2225764 0.68 CDK1 (0.38) CDK1CCNB1CCNA2CCNE1CDK2
SCHEMBL2224393 0.68 NTRK1 (0.45)
SCHEMBL2225236 0.67 TNNI3K (0.51) TNNI3KJAK3CDK1CCNB1CCNA2
SCHEMBL12517788 0.64 TNNI3K (1.00) TNNI3K
SCHEMBL9980493 0.62 TNNI3K (0.36) TNNI3KLRRK2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2523559-A1 COMPOUNDS AND METHODS GlaxoSmithKline LLC (US) 2012-11-21 EP disclosed
WO-2011088027-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2011-07-21 WO disclosed