SCHEMBL2227642

SCHEMBL2227642

O=CCC(F)(F)F.c1ccc2c3c(oc2c1)CNCC3

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 19/20 0.47
KCNH2 Q12809 1/20 0.44
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2226594 0.89 HTR6 (0.46) HTR6KCNH2KDM4EALDH1A1GAA
SCHEMBL171817 0.83 HTR6 (0.58) HTR6KCNH2KDM4E
SCHEMBL30681216 0.83 HTR6 (0.58) HTR6KCNH2KDM4E
Hydrochloric Acid SCHEMBL7140687 0.81 HTR6 (0.59) HTR6KCNH2KDM4E
Isobutyraldehyde SCHEMBL2226850 0.80 HTR6 (0.51) HTR6KCNH2KDM4E
Pentanal SCHEMBL2225046 0.80 HTR6 (0.46) HTR6KCNH2KDM4E
Cyclopentanecarbaldehyde SCHEMBL2229086 0.77 HTR6 (0.48) HTR6KCNH2KDM4E
SCHEMBL2224777 0.75 HTR6 (0.51) HTR6KCNH2
Benzenethiol SCHEMBL2226315 0.75 HTR6 (0.54) HTR6KCNH2KDM4E
SCHEMBL30281730 0.74 HTR6 (0.53) HTR6KCNH2KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011087712-A2 TRICYCLIC DERIVATIVES AND THEIR PHARMACEUTICAL USE AND COMPOSITIONS CEPHALON, INC. (US) 2011-07-21 WO disclosed