SCHEMBL22282192

SCHEMBL22282192

CCCNc1nc(Cl)nc2c1cnn2C[C@H]1O[C@H](CO[Si](C)(C)C(C)(C)C)C2OC(C)(C)O[C@H]21

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SRC P12931 8/20 0.36
ABL1 P00519 7/20 0.36
ALDH1A1 P00352 1/20 0.34
NT5E P21589 8/20 0.34
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
PDE2A O00408 2/20 0.33
ADORA1 P30542 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28599626 1.00 SRC (0.36) SRCABL1ALDH1A1NT5ECYP1A2
SCHEMBL24672311 0.86 NT5E (0.45) NT5E
SCHEMBL28591366 0.85 NT5E (0.44) NT5E
SCHEMBL28610588 0.85 SRC (0.39) SRCABL1ALDH1A1NT5ECYP1A2
SCHEMBL22281833 0.84 NT5E (0.40) SRCABL1NT5E
SCHEMBL22281986 0.84 NT5E (0.40) SRCABL1NT5E
SCHEMBL28610663 0.83 NT5E (0.45) NT5EPDE2A
SCHEMBL28610664 0.83 NT5E (0.45) NT5EPDE2A
SCHEMBL28610592 0.80 NT5E (0.36) NT5E
SCHEMBL28600138 0.74 NT5E (0.48) NT5E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020151707-A1 NOVEL SMALL MOLECULE CD73 INHIBITOR, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL USE THEREOF 江苏恒瑞医药股份有限公司 2020-07-30 WO disclosed