SCHEMBL28610663

SCHEMBL28610663

C[C@H](Nc1nc(Cl)nc2c1cnn2C[C@H]1O[C@H](CO[Si](C)(C)C(C)(C)C)[C@H]2OC(C)(C)O[C@H]21)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NT5E P21589 17/20 0.45
PDE2A O00408 1/20 0.39
KDR P35968 1/20 0.36
PDE9A O76083 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28610664 1.00 NT5E (0.45) NT5EPDE2AKDRPDE9A
SCHEMBL28918241 0.86 NT5E (0.47) NT5EPDE2AKDRPDE9A
SCHEMBL28918240 0.86 NT5E (0.47) NT5EPDE2AKDRPDE9A
SCHEMBL22281832 0.85 NT5E (0.46) NT5EPDE2A
SCHEMBL28595914 0.85 NT5E (0.46) NT5EPDE2A
SCHEMBL28599626 0.83 SRC (0.36) NT5EPDE2A
SCHEMBL22282192 0.83 SRC (0.36) NT5EPDE2A
SCHEMBL24672311 0.82 NT5E (0.45) NT5E
SCHEMBL28591366 0.81 NT5E (0.44) NT5E
SCHEMBL28610592 0.81 NT5E (0.36) NT5E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112955444-A Novel small-molecule CD73 inhibitor, preparation method thereof and application thereof in medicine 江苏恒瑞医药股份有限公司 2021-06-11 CN disclosed