SCHEMBL2228485

SCHEMBL2228485

O=c1c(C=NCCN2CCOCC2)c(NCCN2CCOCC2)nc2ccccn12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.61
ALDH1A1 P00352 7/20 0.61
HSD17B10 Q99714 4/20 0.61
CASP1 P29466 3/20 0.61
CASP7 P55210 3/20 0.61
MEN1 O00255 2/20 0.61
KMT2A Q03164 2/20 0.61
LMNA P02545 2/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
GBA1 P04062 1/20 0.48
RXFP1 Q9HBX9 1/20 0.48
TRIM33 Q9UPN9 2/20 0.47
TRIM24 O15164 1/20 0.47
GAA P10253 4/20 0.47
ADRA1B P35368 1/20 0.47
SALL4 Q9UJQ4 1/20 0.47
HPGD P15428 5/20 0.46
GLA P06280 1/20 0.46
ALOX15 P16050 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2292324 0.91 ALDH1A1 (0.55) KDM4EALDH1A1HSD17B10CASP1CASP7
SCHEMBL2227543 0.80 ALDH1A1 (0.52) KDM4EALDH1A1HSD17B10CASP1CASP7
SCHEMBL12517358 0.78 GBA1 (0.51) KDM4EALDH1A1HSD17B10CASP1CASP7
SCHEMBL2228416 0.77 KDM4E (0.60) KDM4EALDH1A1HSD17B10CASP1CASP7
SCHEMBL2227307 0.77 KDM4E (0.60) KDM4EALDH1A1HSD17B10CASP1CASP7
SCHEMBL12517342 0.77 KDM4E (0.60) KDM4EALDH1A1HSD17B10CASP1CASP7
SCHEMBL12517664 0.77 KDM4E (0.60) KDM4EALDH1A1HSD17B10CASP1CASP7
Hydrochloric Acid SCHEMBL2229679 0.77 GBA1 (0.50) KDM4EALDH1A1HSD17B10CASP1CASP7
SCHEMBL2229506 0.75 KDM4E (0.57) KDM4EALDH1A1HSD17B10CASP1CASP7
SCHEMBL2228471 0.74 KDM4E (0.53) KDM4EALDH1A1HSD17B10CASP1CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011089457-A1 NOVEL MEDICINAL COMPOUNDS URATIM GYÁRTÓ KORLÁTOLT FELELŐSSÉGŰ TÁRSASÁG (HU) 2011-07-28 WO disclosed