SCHEMBL2228946

SCHEMBL2228946

Cc1ccc(S(=O)(=O)OC(=NNc2cccc(C(F)(F)F)c2)C(F)(F)F)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.56
CDK1 P06493 1/20 0.56
CCNB1 P14635 1/20 0.56
CCNA2 P20248 1/20 0.56
CDK2 P24941 1/20 0.56
CDK7 P50613 1/20 0.56
CCNH P51946 1/20 0.56
CCNA1 P78396 1/20 0.56
FFAR4 Q5NUL3 1/20 0.56
MAPT P10636 8/20 0.50
MEN1 O00255 5/20 0.50
KMT2A Q03164 5/20 0.50
LMNA P02545 4/20 0.50
ALOX12 P18054 3/20 0.50
HTT P42858 3/20 0.50
TP53 P04637 2/20 0.50
NPSR1 Q6W5P4 2/20 0.50
POLB P06746 1/20 0.50
XBP1 P17861 1/20 0.50
ALDH1A1 P00352 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2228941 1.00 FFAR1 (0.56) FFAR1CDK1CCNB1CCNA2CDK2
SCHEMBL2228937 1.00 FFAR1 (0.56) FFAR1CDK1CCNB1CCNA2CDK2
SCHEMBL7568797 0.84 P2RY2 (0.42) FFAR1CDK1CCNB1CCNA2CDK2
SCHEMBL7637263 0.84 P2RY2 (0.42) FFAR1CDK1CCNB1CCNA2CDK2
SCHEMBL7569209 0.78 BRD4 (0.43) MAPTLMNAALDH1A1BRD4
SCHEMBL8359192 0.76 PLA2G7 (0.38) MAPTMEN1KMT2ALMNANPSR1
SCHEMBL5441050 0.76 PLA2G7 (0.38) MAPTMEN1KMT2ALMNANPSR1
SCHEMBL23928582 0.71 MEN1 (0.71) FFAR1CDK1CCNB1CCNA2CDK2
SCHEMBL10514960 0.70 MAPT (0.58) MAPTMEN1KMT2ALMNAHTT
SCHEMBL29599829 0.70 MEN1 (0.55) FFAR1CDK1CCNB1CCNA2CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7977358-B2 Pyrazol derivatives HOFFMANN-LA ROCHE INC. (US) 2011-07-12 US disclosed
EP-2182953-A2 NEW PYRAZOL DERIVATIVES F. Hoffmann-Roche AG (CH) 2010-05-12 EP disclosed
WO-2009013211-A2 NEW PYRAZOL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-01-29 WO disclosed