SCHEMBL22296394

SCHEMBL22296394

C=CC(=O)N1CCC2CN(C)CC21

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 9/20 0.40
BTK Q06187 7/20 0.39
JAK3 P52333 2/20 0.38
EGFR P00533 1/20 0.37
SRC P12931 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21186661 0.86 BTK (0.39) HRH3BTK
SCHEMBL21707124 0.79 BTK (0.38) BTKJAK3EGFRSRC
SCHEMBL25558018 0.74 SRC (0.37) BTKJAK3SRC
SCHEMBL4916392 0.72 USP30 (0.42)
SCHEMBL2410020 0.72 USP30 (0.42)
SCHEMBL4916393 0.72 USP30 (0.42)
SCHEMBL22296243 0.72 BTK (0.36) HRH3BTKEGFR
SCHEMBL22296241 0.71 HRH3 (0.40) HRH3
SCHEMBL30231523 0.70 PARP1 (0.36) HRH3BTKJAK3SRC
SCHEMBL22881068 0.70 SRC (0.33) JAK3SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3689871-A1 4,6,7-TRISUBSTITUTED 1,2-DIHYDROPYRROL[3,4-C]PYRIDIN/PYRIMIDIN-3-ONE DERIVATIVE AND USE Shanghai Haiyan Pharmaceutical Technology Co., Ltd. (CN) 2020-08-05 EP disclosed