SCHEMBL22296830

SCHEMBL22296830

COC(=O)C[C@@]1(c2ccccn2)CCOC2(CCCC2)C1

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 20/20 0.60
OPRD1 P41143 2/20 0.58
OPRK1 P41145 2/20 0.58
KCNH2 Q12809 2/20 0.58
SCN5A Q14524 2/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2D6 P10635 1/20 0.58
DRD2 P14416 1/20 0.58
DRD3 P35462 1/20 0.58
CACNA1C Q13936 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22296894 1.00 OPRM1 (0.60) OPRM1OPRD1OPRK1KCNH2SCN5A
SCHEMBL26638645 0.89 OPRM1 (0.56) OPRM1OPRD1OPRK1KCNH2SCN5A
SCHEMBL29808298 0.86 OPRM1 (0.64) OPRM1OPRD1OPRK1KCNH2SCN5A
SCHEMBL22283293 0.86 OPRM1 (0.64) OPRM1OPRD1OPRK1KCNH2SCN5A
SCHEMBL30288497 0.86 OPRM1 (0.64) OPRM1OPRD1OPRK1KCNH2SCN5A
SCHEMBL22261623 0.86 OPRM1 (0.64) OPRM1OPRD1OPRK1KCNH2SCN5A
SCHEMBL22296825 0.85 OPRM1 (0.54) OPRM1OPRD1OPRK1KCNH2SCN5A
SCHEMBL29967521 0.82 OPRM1 (0.65) OPRM1OPRD1OPRK1KCNH2SCN5A
SCHEMBL26638893 0.82 OPRM1 (0.65) OPRM1OPRD1OPRK1KCNH2SCN5A
SCHEMBL30286713 0.81 OPRM1 (0.70) OPRM1OPRD1OPRK1KCNH2SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4265604-A1 OXASPIRO SUBSTITUTED PYRROLOPYRAZOLE DERIVATIVE, INTERMEDIATE THEREOF, AND PREPARATION METHOD THEREFOR Shanghai Haiyan Pharmaceutical Technology Co., Ltd (CN) 2023-10-25 EP disclosed
EP-3689859-A1 METHOD FOR PREPARING OXASPIROCYCLE DERIVATIVE, AND INTERMEDIATE THEREOF Jiangsu Hengrui Medicine Co., Ltd. (CN) 2020-08-05 EP disclosed