SCHEMBL22297464

SCHEMBL22297464

FC(F)(F)C(F)(c1ccc2c(c1)CCC1CCC[C@@H]21)C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SRD5A1 P18405 1/20 0.40
HSD17B1 P14061 2/20 0.34
RORC P51449 8/20 0.34
STS P08842 3/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA5A P35218 1/20 0.34
CA9 Q16790 1/20 0.34
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
SIGMAR1 Q99720 4/20 0.33
PNMT P11086 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22297755 1.00 SRD5A1 (0.40) SRD5A1HSD17B1RORCSTSCA1
SCHEMBL20153507 1.00 SRD5A1 (0.40) SRD5A1HSD17B1RORCSTSCA1
SCHEMBL20153523 1.00 SRD5A1 (0.40) SRD5A1HSD17B1RORCSTSCA1
SCHEMBL20153589 0.94 SRD5A1 (0.38) SRD5A1RORCSTSCA1CA2
SCHEMBL20153556 0.86 SRD5A1 (0.41) SRD5A1HSD17B1STSCA1CA2
SCHEMBL23677460 0.74 SRD5A1 (0.39) SRD5A1RORCSTSCA1CA2
SCHEMBL22297799 0.74 STS (0.42) SRD5A1RORCSTSCA1CA2
SCHEMBL22297451 0.74 AR (0.49) RORCNOS3NOS1NOS2PNMT
SCHEMBL20153520 0.74 AR (0.49) RORCNOS3NOS1NOS2PNMT
SCHEMBL20068379 0.74 SRD5A1 (0.39) SRD5A1RORCSTSCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3541786-B1 TRICYCLIC SULFONES AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2020-08-05 EP disclosed