SCHEMBL2230092

SCHEMBL2230092

CC1=CC(=O)N(c2cc(N3C(=O)C=CC3=O)ccc2C)C1=O

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 12/20 0.44
HSP90AA1 P07900 4/20 0.44
G6PD P11413 2/20 0.43
TLR9 Q9NR96 1/20 0.43
FAAH O00519 3/20 0.42
CCR6 P51684 3/20 0.41
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
PKM P14618 1/20 0.39
HPGD P15428 1/20 0.39
MCL1 Q07820 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2228521 0.94 MGLL (0.46) MGLLHSP90AA1G6PDTLR9FAAH
SCHEMBL1116215 0.92 KMT2A (0.41) MGLLHSP90AA1G6PDTLR9MEN1
SCHEMBL94095 0.85 MGLL (0.57) MGLLHSP90AA1G6PDTLR9FAAH
SCHEMBL4839640 0.81 MGLL (0.61) MGLLHSP90AA1FAAHCCR6ALDH1A1
SCHEMBL2229875 0.80 MGLL (0.43) MGLLHSP90AA1G6PDTLR9FAAH
SCHEMBL3686454 0.79 KMT2A (0.41) MGLLHSP90AA1G6PDTLR9MEN1
SCHEMBL21409967 0.79 MGLL (0.66) MGLLHSP90AA1G6PDTLR9FAAH
SCHEMBL20385941 0.78 CCR6 (0.55) MGLLHSP90AA1G6PDFAAHCCR6
SCHEMBL23442665 0.78 MGLL (0.47) MGLLHSP90AA1G6PDTLR9FAAH
SCHEMBL3684376 0.77 HPGD (0.34) MGLLHSP90AA1CCR6ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11230636-B2 Rubber composition having improved properties in the raw state and in the cooked state COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2022-01-25 US claimed
EP-3582977-B1 RUBBER COMPOSITION HAVING IMPROVED PROPERTIES IN THE RAW STATE AND IN THE COOKED STATE MICHELIN & CIE (FR) 2021-03-31 EP claimed
US-20200056017-A1 RUBBER COMPOSITION HAVING IMPROVED PROPERTIES IN THE RAW STATE AND IN THE COOKED STATE COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2020-02-20 US claimed
WO-2018150136-A1 RUBBER COMPOSITION HAVING IMPROVED PROPERTIES IN THE RAW STATE AND IN THE COOKED STATE COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2018-08-23 WO claimed
JP-4717814-B2 2011-07-06 JP claimed
US-7442733-B2 Rubber composition comprising a citraconimidomaleimide MICHELIN RECHERCHE ET TECHNIQUE S.A. (CH) 2008-10-28 US claimed
US-20060247342-A1 Rubber composition comprising a citraconimidomaleimide MICHELIN RECHERCHE ET TECHNIQUE S.A. 2006-11-02 US claimed
EP-1664180-A1 RUBBER COMPOSITION COMPRISING A CITRACONIMIDO-MALEIMIDE Société de Technologie Michelin (FR) 2006-06-07 EP claimed
WO-2005026250-A1 RUBBER COMPOSITION COMPRISING A CITRACONIMIDO-MALEIMIDE SOCIETE DE TECHNOLOGIE MICHELIN (FR) 2005-03-24 WO claimed
US-11230636-B2 Rubber composition having improved properties in the raw state and in the cooked state COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2022-01-25 US disclosed
EP-3582977-B1 RUBBER COMPOSITION HAVING IMPROVED PROPERTIES IN THE RAW STATE AND IN THE COOKED STATE MICHELIN & CIE (FR) 2021-03-31 EP disclosed
US-20200056017-A1 RUBBER COMPOSITION HAVING IMPROVED PROPERTIES IN THE RAW STATE AND IN THE COOKED STATE COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2020-02-20 US disclosed
WO-2018150136-A1 RUBBER COMPOSITION HAVING IMPROVED PROPERTIES IN THE RAW STATE AND IN THE COOKED STATE COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2018-08-23 WO disclosed
US-7442733-B2 Rubber composition comprising a citraconimidomaleimide MICHELIN RECHERCHE ET TECHNIQUE S.A. (CH) 2008-10-28 US disclosed
US-20060247342-A1 Rubber composition comprising a citraconimidomaleimide MICHELIN RECHERCHE ET TECHNIQUE S.A. 2006-11-02 US disclosed
EP-1664180-A1 RUBBER COMPOSITION COMPRISING A CITRACONIMIDO-MALEIMIDE Société de Technologie Michelin (FR) 2006-06-07 EP disclosed
WO-2005026250-A1 RUBBER COMPOSITION COMPRISING A CITRACONIMIDO-MALEIMIDE SOCIETE DE TECHNOLOGIE MICHELIN (FR) 2005-03-24 WO disclosed