SCHEMBL22304487

SCHEMBL22304487

CCOC(=O)c1cccc(CN2CC3(COC3)C2)n1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.52
MAPT P10636 1/20 0.44
PDCD1 Q15116 1/20 0.42
CD274 Q9NZQ7 1/20 0.42
PFKFB3 Q16875 1/20 0.41
GAA P10253 1/20 0.40
ALDH1A1 P00352 5/20 0.36
KDM4E B2RXH2 3/20 0.36
GABRA2 P47869 1/20 0.36
GABRB2 P47870 1/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CXCR4 P61073 1/20 0.36
NTRK1 P04629 1/20 0.36
TP53 P04637 1/20 0.35
POLB P06746 2/20 0.35
MAPK1 P28482 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1811182 0.81 CYP1A2 (0.55) CYP1A2MAPTPFKFB3GAAALDH1A1
SCHEMBL31186040 0.77 CYP1A2 (0.56) CYP1A2MAPTGAAALDH1A1KDM4E
SCHEMBL2822250 0.76 CYP1A2 (0.55) CYP1A2MAPTGAAALDH1A1KDM4E
SCHEMBL2817557 0.76 CYP1A2 (0.55) CYP1A2MAPTGAAALDH1A1KDM4E
SCHEMBL31186092 0.76 CYP1A2 (0.51) CYP1A2MAPTGAAALDH1A1KDM4E
SCHEMBL22304530 0.74 CYP1A2 (0.52) CYP1A2MAPTPFKFB3GAAALDH1A1
SCHEMBL30080477 0.74 CXCR4 (0.49) PDCD1CD274CXCR4NTRK1
SCHEMBL31186103 0.74 CYP1A2 (0.49) CYP1A2MAPTGAAALDH1A1KDM4E
SCHEMBL7336055 0.74 CYP1A2 (0.77) CYP1A2MAPTGAAALDH1A1KDM4E
SCHEMBL536661 0.72 CYP1A2 (0.74) CYP1A2MAPTGAAALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112996783-B 2-aminopyrimidine derivatives, preparation method and application thereof in medicines 江苏恒瑞医药股份有限公司 2022-11-18 CN disclosed
WO-2020156505-A1 2-AMIONPYRIMIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF IN MEDICINES 江苏恒瑞医药股份有限公司 2020-08-06 WO disclosed