SCHEMBL22304530

SCHEMBL22304530

CCOC(=O)c1cccc(N2CCC3(CC2)COC3)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.52
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
KDM4E B2RXH2 2/20 0.45
RXFP1 Q9HBX9 1/20 0.45
KIF18A Q8NI77 5/20 0.45
MAPT P10636 1/20 0.44
KMT2A Q03164 1/20 0.44
CRBN Q96SW2 1/20 0.43
PIK3CA P42336 1/20 0.41
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
HSD17B10 Q99714 1/20 0.40
IRAK4 Q9NWZ3 1/20 0.39
PFKFB3 Q16875 1/20 0.39
GABRA2 P47869 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1811182 0.88 CYP1A2 (0.55) CYP1A2NPC1RAB9AKDM4ERXFP1
SCHEMBL30080383 0.87 CRBN (0.55) CYP1A2KIF18AKMT2ACRBNALDH1A1
SCHEMBL31337804 0.84 CYP1A2 (0.56) CYP1A2NPC1RAB9AKDM4ERXFP1
SCHEMBL2810512 0.84 CYP1A2 (0.59) CYP1A2NPC1RAB9AKDM4ERXFP1
SCHEMBL22304477 0.81 CYP1A2 (0.52) CYP1A2NPC1RAB9AKDM4ERXFP1
SCHEMBL21875248 0.81 CYP1A2 (0.62) CYP1A2NPC1RAB9AKDM4ERXFP1
SCHEMBL28534611 0.80 CYP1A2 (0.60) CYP1A2NPC1RAB9AKDM4ERXFP1
SCHEMBL6967592 0.79 CYP1A2 (0.59) CYP1A2NPC1RAB9AKDM4ERXFP1
SCHEMBL441409 0.78 CYP1A2 (0.57) CYP1A2NPC1RAB9AKDM4ERXFP1
Hydrochloric Acid SCHEMBL445411 0.78 CYP1A2 (0.57) CYP1A2NPC1RAB9AKDM4ERXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020156505-A1 2-AMIONPYRIMIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF IN MEDICINES 江苏恒瑞医药股份有限公司 2020-08-06 WO disclosed