SCHEMBL22309130

SCHEMBL22309130

CC(=O)c1ccc(-c2ccc(F)cc2)nc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.73
RXFP1 Q9HBX9 2/20 0.73
PTPN1 P18031 1/20 0.59
PTPN6 P29350 1/20 0.59
PTPN11 Q06124 1/20 0.59
LDHA P00338 2/20 0.50
FYN P06241 1/20 0.49
ALOX5 P09917 1/20 0.48
HPGDS O60760 1/20 0.48
BAZ2B Q9UIF8 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.46
RAB9A P51151 2/20 0.46
DGAT1 O75907 1/20 0.46
HDAC2 Q92769 1/20 0.45
PTGS1 P23219 1/20 0.45
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
KMT2A Q03164 1/20 0.44
TP53 P04637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30436727 1.00 NPC1 (0.73) NPC1RXFP1PTPN1PTPN6PTPN11
SCHEMBL3502067 0.90 NPC1 (0.63) NPC1RXFP1PTPN1PTPN6PTPN11
SCHEMBL12436558 0.89 LDHA (0.56) NPC1RXFP1PTPN1PTPN6PTPN11
SCHEMBL2947695 0.84 NPC1 (0.75) NPC1RXFP1PTPN1PTPN6PTPN11
SCHEMBL16991665 0.84 NPC1 (0.51) NPC1RXFP1LDHABAZ2BSMN1; SMN2
SCHEMBL12392719 0.84 LDHA (0.66) NPC1RXFP1LDHAHPGDSBAZ2B
SCHEMBL2343432 0.83 LDHA (0.64) NPC1RXFP1LDHAHPGDSBAZ2B
SCHEMBL2343427 0.83 LDHA (0.64) NPC1RXFP1LDHAHPGDSBAZ2B
SCHEMBL5658059 0.83 RXFP1 (0.73) NPC1RXFP1PTPN1PTPN6PTPN11
SCHEMBL13100100 0.82 LDHA (0.73) NPC1RXFP1PTPN1LDHAHPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111499613-B N-carboxamide derivatives, method for the production thereof and their use in medicine 浙江海正药业股份有限公司 2023-05-12 CN disclosed
CN-111499613-A N-formamide derivative, preparation method and medical application thereof 浙江海正药业股份有限公司 2020-08-07 CN disclosed
WO-2020156319-A1 N-FORMAMIDE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 浙江海正药业股份有限公司 2020-08-06 WO disclosed