SCHEMBL22312949

SCHEMBL22312949

C=CCCC(=O)C(C[C@H](C)N(C)C)(c1ccccc1)c1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 6/20 0.67
GRIN2A Q12879 6/20 0.67
GRIN2D O15399 5/20 0.67
GRIN2C Q14957 5/20 0.67
GRIN2B Q13224 4/20 0.67
OPRM1 P35372 4/20 0.67
KCNH2 Q12809 3/20 0.67
DRD3 P35462 3/20 0.67
DRD4 P21917 2/20 0.67
CACNA1F O60840 1/20 0.67
ABCB1 P08183 1/20 0.67
CYP2B6 P20813 1/20 0.67
OPRD1 P41143 1/20 0.67
OPRK1 P41145 1/20 0.67
CACNA1D Q01668 1/20 0.67
CACNA1S Q13698 1/20 0.67
CACNA1C Q13936 1/20 0.67
MRGPRX2 Q96LB1 1/20 0.67
DRD2 P14416 1/20 0.40
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8661873 0.92 GRIN1 (0.64) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B
SCHEMBL3166469 0.88 GRIN1 (0.68) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B
SCHEMBL22312261 0.86 GRIN1 (0.70) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B
SCHEMBL22312943 0.82 GRIN1 (0.72) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B
SCHEMBL22312251 0.81 GRIN1 (0.70) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B
SCHEMBL11312228 0.81 GRIN1 (0.70) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B
SCHEMBL22312256 0.81 GRIN1 (0.74) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B
Methadone SCHEMBL28890984 0.81 GRIN1 (0.94) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B
SCHEMBL22312956 0.81 GRIN1 (0.65) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B
Methadone SCHEMBL34140 0.80 GRIN1 (1.00) GRIN1GRIN2AGRIN2DGRIN2CGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020159587-A1 STRUCTURALLY MODIFIED OPIOIDS FOR PREVENTION AND TREATMENT OF DISEASES AND CONDITIONS UNIVERSITY OF PADOVA (IT) 2020-08-06 WO disclosed