SCHEMBL223209

SCHEMBL223209

Nc1ccn([C@@H]2O[C@H](C(O)F)[C@@H](O)[C@H]2O)c(=O)n1

nearest known ligand 0.65

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NT5E P21589 1/20 0.65
LMNA P02545 1/20 0.62
THRB P10828 1/20 0.62
MTOR P42345 1/20 0.62
MDM2 Q00987 1/20 0.62
NCOA1 Q15788 1/20 0.62
NCOA3 Q9Y6Q9 1/20 0.62
PDE4D Q08499 1/20 0.46
PDE3A Q14432 1/20 0.46
SLC29A1 Q99808 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
ST6GAL1 P15907 3/20 0.44
TSHR P16473 1/20 0.44
GLA P06280 1/20 0.44
P2RY2 P41231 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6312068 1.00 NT5E (0.65) NT5ELMNATHRBMTORMDM2
SCHEMBL4414290 0.88 NT5E (0.67) NT5ELMNATHRBMTORMDM2
SCHEMBL800348 0.87 NT5E (0.65) NT5ELMNATHRBMTORMDM2
SCHEMBL13190277 0.87 NT5E (0.65) NT5ELMNATHRBMTORMDM2
SCHEMBL800434 0.87 NT5E (0.65) NT5ELMNATHRBMTORMDM2
SCHEMBL4946500 0.87 NT5E (0.65) NT5ELMNATHRBMTORMDM2
SCHEMBL7539957 0.87 NT5E (0.65) NT5ELMNATHRBMTORMDM2
SCHEMBL800395 0.87 NT5E (0.65) NT5ELMNATHRBMTORMDM2
SCHEMBL13134657 0.87 NT5E (0.65) NT5ELMNATHRBMTORMDM2
SCHEMBL452913 0.87 NT5E (0.65) NT5ELMNATHRBMTORMDM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 750 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116333019-B Fluorocytidine compound and preparation method and application thereof 沈阳农业大学 2024-04-02 CN claimed
WO-2023150622-A2 RNAI AGENTS FOR INHIBITING EXPRESSION OF CORONAVIRUS (COV) VIRAL GENOMES, COMPOSITIONS THEREOF, AND METHODS OF USE Arrowhead Pharmaceuticals, Inc. (US) 2023-08-10 WO claimed
CN-116333019-A Fluorocytidine compound and preparation method and application thereof 沈阳农业大学 2023-06-27 CN claimed
WO-2019195494-A1 COMPOSITIONS AND METHODS FOR SYNTHESIS OF PHOSPHORYLATED MOLECULES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-10-10 WO claimed
US-20190292540-A1 SPINAL MUSCULAR ATROPHY (SMA) TREATMENT VIA TARGETING OF SMN2 SPLICE SITE INHIBITORY SEQUENCES UNIV MASSACHUSETTS (US) 2019-09-26 US claimed
US-20170096664-A1 SPINAL MUSCULAR ATROPHY (SMA) TREATMENT VIA TARGETING OF SMN2 SPLICE SITE INHIBITORY SEQUENCES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2017-04-06 US claimed
US-9260760-B2 Method for determining complete response to anticancer therapy BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2016-02-16 US claimed
US-20150152504-A1 METHOD FOR DETERMINING COMPLETE RESPONSE TO ANTICANCER THERAPY BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2015-06-04 US claimed
US-8889645-B2 Nucleic acid modulators of glycoprotein VI REGADO BIOSCIENCES, INC. (US) 2014-11-18 US claimed
US-20140128587-A1 NUCLEIC ACID MODULATORS OF GLYCOPROTEIN VI REGADO BIOSCIENCES, INC. (US) 2014-05-08 US claimed
EP-0504279-B1 FERMENTATION PROCESS FOR THE PRODUCTION OF PYRIMIDINE DEOXYRIBONUCLEOSIDES CHEMGEN CORP (US) 1997-07-09 EP claimed
US-5476932-A Process for producing N4-acyl-5'-deoxy-5-fluorocytidine derivatives HOFFMANN-LA ROCHE INC. (US) 1995-12-19 US claimed
US-5453497-A Process for producing N4 -acyl-5'-deoxy-5-fluorocytidine compounds HOFFMANN-LA ROCHE INC. (US) 1995-09-26 US claimed
EP-0637966-A1 BYSTANDER EFFECT TUMORICIDAL THERAPY. US HEALTH (US) 1995-02-15 EP claimed
WO-1993021959-A1 BYSTANDER EFFECT TUMORICIDAL THERAPY THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1993-11-11 WO claimed
US-5213972-A Production of thymidine and deoxyuridine, intermediates for AZT CHEMGEN CORPORATION (US) 1993-05-25 US claimed
EP-0504279-A4 FERMENTATION PROCESS FOR THE PRODUCTION OF PYRIMIDINE DEOXYRIBONUCLEOSIDES 1993-02-17 EP claimed
EP-0504279-A1 FERMENTATION PROCESS FOR THE PRODUCTION OF PYRIMIDINE DEOXYRIBONUCLEOSIDES. CHEMGEN CORP (US) 1992-09-23 EP claimed
WO-1991009130-A1 FERMENTATION PROCESS FOR THE PRODUCTION OF PYRIMIDINE DEOXYRIBONUCLEOSIDES CHEMGEN CORPORATION (US) 1991-06-27 WO claimed
CN-1045791-A Use the cooperative compositions HIV inhibiting of nucleoside derivates ONCOGEN (US) 1990-10-03 CN claimed