SCHEMBL2232358

SCHEMBL2232358

Cc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccc3)C2c2ccc(C(C)C)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 6/20 0.59
CCR2 P41597 2/20 0.54
KDM4E B2RXH2 3/20 0.52
HPGD P15428 1/20 0.52
RXFP1 Q9HBX9 4/20 0.51
ANXA2 P07355 4/20 0.50
S100A10 P60903 4/20 0.50
MEN1 O00255 4/20 0.49
KMT2A Q03164 4/20 0.49
P2RX3 P56373 2/20 0.49
CRHBP P24387 1/20 0.49
CRHR2 Q13324 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
LMNA P02545 1/20 0.49
TP53 P04637 1/20 0.47
ALDH1A1 P00352 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12943495 0.88 ALDH1A1 (0.59) CCR1CCR2KDM4EHPGDRXFP1
SCHEMBL2232399 0.86 CCR1 (0.54) CCR1CCR2KDM4EHPGDRXFP1
SCHEMBL8776139 0.85 RXFP1 (0.55) CCR1KDM4EHPGDRXFP1ANXA2
SCHEMBL12943493 0.85 RXFP1 (0.63) CCR1CCR2KDM4EHPGDRXFP1
SCHEMBL934299 0.84 CCR1 (0.51) CCR1CCR2KDM4ERXFP1ANXA2
SCHEMBL16370574 0.82 GAA (0.64) CCR1CCR2KDM4EHPGDRXFP1
SCHEMBL6115917 0.82 RXFP1 (0.55) CCR1CCR2KDM4ERXFP1ANXA2
SCHEMBL10146036 0.82 RXFP1 (0.69) CCR1CCR2KDM4EHPGDRXFP1
SCHEMBL6116449 0.82 RXFP1 (0.54) CCR1CCR2KDM4ERXFP1ANXA2
SCHEMBL934178 0.81 RXFP1 (0.52) CCR1CCR2KDM4ERXFP1ANXA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011092505-A1 S100 PROTEIN BINDING INTERACTION INHIBITORS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2011-08-04 WO claimed
WO-2011092505-A1 S100 PROTEIN BINDING INTERACTION INHIBITORS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2011-08-04 WO disclosed