SCHEMBL22325264

SCHEMBL22325264

COC(Cc1c(Cl)ncnc1Cl)OC

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
LMNA P02545 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
ENPP1 P22413 2/20 0.33
CYP2C9 P11712 1/20 0.33
HPGD P15428 1/20 0.33
CYP2C19 P33261 1/20 0.33
AURKA O14965 1/20 0.30
POLB P06746 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
SELE P16581 1/20 0.30
VCAM1 P19320 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22325322 0.87 ALDH1A1 (0.39) ALDH1A1LMNASMN1; SMN2
SCHEMBL1795269 0.80 ALDH1A1 (0.39) ALDH1A1LMNASMN1; SMN2ENPP1SELE
SCHEMBL22325329 0.78 ALDH1A1 (0.33) ALDH1A1LMNASMN1; SMN2
SCHEMBL2231346 0.76 ALDH1A1 (0.40) ALDH1A1LMNASMN1; SMN2POLBSELE
SCHEMBL8323588 0.75 ALDH1A1 (0.46) ALDH1A1LMNASMN1; SMN2CYP2C9HPGD
SCHEMBL22343500 0.73 ATR (0.42) AURKAPOLB
SCHEMBL22343501 0.73 PDPK1 (0.39) ALDH1A1LMNASMN1; SMN2
SCHEMBL28681146 0.72
SCHEMBL22308707 0.71 ALDH1A1 (0.38) ALDH1A1LMNASMN1; SMN2CYP2C9CYP2C19
SCHEMBL10249025 0.71 ALDH1A1 (0.38) ALDH1A1LMNASMN1; SMN2ENPP1SELE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12325707-B2 Process for preparing enantiomerically enriched JAK inhibitors SUN PHARMACEUTICAL INDUSTRIES, INC. (US) 2025-06-10 US disclosed
US-20240368166-A1 PROCESS FOR PREPARING ENANTIOMERICALLY ENRICHED JAK INHIBITORS SUN PHARMACEUTICAL INDUSTRIES, INC. 2024-11-07 US disclosed
US-20240300963-A1 PROCESS FOR PREPARING ENANTIOMERICALLY ENRICHED JAK INHIBITORS SUN PHARMACEUTICAL INDUSTRIES, INC. 2024-09-12 US disclosed
WO-2023018954-A1 TREATMENT OF JAK-INHIBITION-RESPONSIVE DISORDERS WITH PRODRUGS OF JAK INHIBITORS CONCERT PHARMACEUTICALS, INC. (US) 2023-02-16 WO disclosed
US-20220306636-A1 PROCESS FOR PREPARING ENANTIOMERICALLY ENRICHED JAK INHIBITORS SUN PHARMACEUTICAL INDUSTRIES, INC. 2022-09-29 US disclosed
US-20220213105-A1 PROCESS FOR PREPARING ENANTIOMERICALLY ENRICHED JAK INHIBITORS SUN PHARMACEUTICAL INDUSTRIES, INC. 2022-07-07 US disclosed
US-20220213105-A1 PROCESS FOR PREPARING ENANTIOMERICALLY ENRICHED JAK INHIBITORS SUN PHARMACEUTICAL INDUSTRIES, INC. 2022-07-07 US disclosed
CN-113906032-A Methods for preparing enantiomerically enriched JAK inhibitors 康塞特医药品有限公司 2022-01-07 CN disclosed
EP-3921318-A1 PROCESS FOR PREPARING ENANTIOMERICALLY ENRICHED JAK INHIBITORS Concert Pharmaceuticals Inc. (US) 2021-12-15 EP disclosed
WO-2020163653-A1 PROCESS FOR PREPARING ENANTIOMERICALLY ENRICHED JAK INHIBITORS CONCERT PHARMACEUTICALS, INC. (US) 2020-08-13 WO disclosed
WO-2020163653-A1 PROCESS FOR PREPARING ENANTIOMERICALLY ENRICHED JAK INHIBITORS CONCERT PHARMACEUTICALS, INC. (US) 2020-08-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12325707-B2 Process for preparing enantiomerically enriched JAK inhibitors JAK1, JAK2, JAK3 ALDH1A1 2401/4885LMNA 4673/4885SMN1; SMN2 4541/4885
US-20220213105-A1 PROCESS FOR PREPARING ENANTIOMERICALLY ENRICHED JAK INHIBITORS JAK1, JAK2, JAK3 ALDH1A1 2401/4885LMNA 4673/4885SMN1; SMN2 4541/4885
US-20240300963-A1 PROCESS FOR PREPARING ENANTIOMERICALLY ENRICHED JAK INHIBITORS JAK1, JAK2, JAK3 ALDH1A1 2401/4885LMNA 4673/4885SMN1; SMN2 4541/4885
US-20240368166-A1 PROCESS FOR PREPARING ENANTIOMERICALLY ENRICHED JAK INHIBITORS JAK1, JAK2, JAK3 ALDH1A1 2401/4885LMNA 4673/4885SMN1; SMN2 4541/4885
US-20220306636-A1 PROCESS FOR PREPARING ENANTIOMERICALLY ENRICHED JAK INHIBITORS JAK1, JAK2, JAK3 ALDH1A1 2401/4885LMNA 4673/4885SMN1; SMN2 4541/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.