SCHEMBL22328136

SCHEMBL22328136

NC(=O)CN1C[C@H](Cc2ccccc2)NC(=O)CN(C(=O)CCC(=O)O)C[C@H](CCC(=O)O)NC(=O)CN(C(=O)Cc2ccc3c(c2)OCO3)C[C@H](CCC(=O)O)NC(=O)CN(C(=O)CCC2CCCCC2)C[C@H](Cc2ccccc2)NC(=O)c2ccc(cc2)SCCCC1=O

nearest known ligand 0.84

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EPHA2 P29317 2/20 0.84
EGFR P00533 2/20 0.63
NFKBIA P25963 1/20 0.54
AKT1 P31749 1/20 0.54
PTGER2 P43116 2/20 0.42
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
USP19 O94966 1/20 0.31
CNR1 P21554 1/20 0.30
ITGB3 P05106 2/20 0.30
ITGA2B P08514 2/20 0.30
F2R P25116 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22328117 0.91 EPHA2 (1.00) EPHA2EGFRNFKBIAAKT1PTGER2
SCHEMBL19003322 0.77 EPHA2 (0.75) EPHA2EGFRNFKBIAAKT1PTGER2
SCHEMBL19003321 0.77 EPHA2 (0.75) EPHA2EGFRNFKBIAAKT1PTGER2
SCHEMBL22328134 0.72 EPHA2 (1.00) EPHA2EGFRNFKBIAAKT1PTGER2
SCHEMBL24996897 0.71 EGFR (0.87) EPHA2EGFRNFKBIAAKT1PTGER2
SCHEMBL22730944 0.71 EPHA2 (0.65) EPHA2EGFRNFKBIAAKT1PTGER2
SCHEMBL24996893 0.71 EGFR (0.86) EPHA2EGFRNFKBIAAKT1PTGER2
SCHEMBL19003382 0.70 EPHA2 (0.66) EPHA2EGFRNFKBIAAKT1PTGER2
SCHEMBL19003412 0.67 EPHA2 (0.62) EPHA2EGFRNFKBIAAKT1PTGER2
SCHEMBL19003318 0.67 EPHA2 (0.62) EPHA2EGFRNFKBIAAKT1PTGER2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10738082-B2 One-bead-two-compound macrocyclic library and methods of preparation and use UNIVERSITY OF SOUTH FLORIDA (US) 2020-08-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10738082-B2 One-bead-two-compound macrocyclic library and methods of preparation and use EPHA2, EPHA1, EPHB2 EPHA2 1/4885EGFR 26/4885NFKBIA 3054/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.