SCHEMBL2233779

SCHEMBL2233779

COCNS(=O)(=O)c1cccc(C(F)(F)F)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.59
CA2 P00918 1/20 0.59
MMP1 P03956 1/20 0.59
MMP2 P08253 1/20 0.59
MMP9 P14780 1/20 0.59
MMP8 P22894 1/20 0.59
MMP13 P45452 1/20 0.59
TSHR P16473 2/20 0.52
MMP7 P09237 1/20 0.52
ALDH1A1 P00352 2/20 0.51
MAPT P10636 3/20 0.50
KDM4E B2RXH2 2/20 0.50
GAA P10253 2/20 0.50
ALOX15 P16050 2/20 0.50
NR3C1 P04150 1/20 0.50
PGR P06401 1/20 0.50
AR P10275 1/20 0.50
ESR2 Q92731 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29888356 1.00 CA1 (0.59) CA1CA2MMP1MMP2MMP9
SCHEMBL13753685 0.83 CA1 (0.64) CA1CA2MMP1MMP2MMP9
SCHEMBL5189385 0.80 CA1 (0.64) CA1CA2MMP1MMP2MMP9
SCHEMBL4818983 0.79 CA1 (0.59) CA1CA2MMP1MMP2MMP9
SCHEMBL3277623 0.78 TRPV1 (0.58) CA1CA2MMP1MMP2MMP9
SCHEMBL5184452 0.78 CA1 (0.70) CA1CA2MMP1MMP2MMP9
SCHEMBL1148961 0.78 CA1 (0.60) CA1CA2MMP1MMP2MMP9
SCHEMBL29537299 0.77 CA1 (0.74) CA1CA2MMP1MMP2MMP9
SCHEMBL12541679 0.77 CA1 (0.56) CA1CA2MMP1MMP2MMP9
SCHEMBL745591 0.77 ALDH1A1 (0.64) CA1CA2MMP1MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2354126-A1 Heteroaryl sulfonamides and CCR2 ChemoCentryx, Inc. (US) 2011-08-10 EP disclosed
WO-2008008431-A2 HETEROARYL SULFONAMIDES AND CCR2/CCR9 CHEMOCENTRYX, INC. (US) 2008-01-17 WO disclosed