SCHEMBL22353604

SCHEMBL22353604

O=C(O)C1CCC2(CNc3cncc(Br)c3)CCCC1C2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
RXFP1 Q9HBX9 1/20 0.33
L3MBTL1 Q9Y468 3/20 0.32
GRK2 P25098 1/20 0.32
CASP6 P55212 1/20 0.32
CASP8 Q14790 1/20 0.32
CTDSP1 Q9GZU7 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
CXCR3 P49682 1/20 0.32
LMNA P02545 2/20 0.32
SMN1; SMN2 Q16637 3/20 0.31
TAS1R3 Q7RTX0 2/20 0.31
TAS1R1 Q7RTX1 2/20 0.31
TAS1R2 Q8TE23 2/20 0.31
L3MBTL4 Q8NA19 1/20 0.31
L3MBTL3 Q96JM7 1/20 0.31
NPC1 O15118 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22353981 0.85
SCHEMBL22347350 0.74 POLB (0.37) ALDH1A1KDM4EMEN1KMT2AL3MBTL1
SCHEMBL22353654 0.69 SLC9A1 (0.32) ALDH1A1KDM4EPOLB
SCHEMBL22347182 0.69 KDM4E (0.39) ALDH1A1KDM4EMEN1KMT2AL3MBTL1
SCHEMBL3145935 0.67 POLB (0.37) ALDH1A1KDM4EMEN1KMT2AL3MBTL1
SCHEMBL22354081 0.67 KDM4E (0.35) ALDH1A1KDM4EMEN1KMT2AL3MBTL1
SCHEMBL3145942 0.65 HTT (0.38) ALDH1A1KDM4EMEN1KMT2AL3MBTL1
SCHEMBL22347208 0.63
SCHEMBL22353949 0.63
SCHEMBL3773545 0.62 SMN1; SMN2 (0.33) ALDH1A1KDM4ECXCR3SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020168143-A1 SUBSTITUTED BICYCLIC COMPOUNDS AS FARNESOID X RECEPTOR MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2020-08-20 WO disclosed