SCHEMBL22355459

SCHEMBL22355459

CC1CNCc2nc(O)ccc2O1

nearest known ligand 0.35

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.35
BRD4 O60885 1/20 0.31
CREBBP Q92793 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22355454 1.00 NTRK1 (0.35) NTRK1BRD4CREBBP
SCHEMBL22355519 1.00 NTRK1 (0.35) NTRK1BRD4CREBBP
Hydrochloric Acid SCHEMBL26618555 0.98 NTRK1 (0.34) NTRK1BRD4CREBBP
Hydrochloric Acid SCHEMBL30850013 0.98 NTRK1 (0.34) NTRK1BRD4CREBBP
Hydrochloric Acid SCHEMBL29694249 0.98 NTRK1 (0.34) NTRK1BRD4CREBBP
SCHEMBL22355411 0.80 OPRM1 (0.30)
SCHEMBL22355412 0.80 OPRM1 (0.30)
SCHEMBL22355462 0.80 KDM4E (0.30)
SCHEMBL22355524 0.80 OPRM1 (0.30)
SCHEMBL22355460 0.80 KDM4E (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020165776-A1 HYDROXYPYRIDOXAZEPINES AS NRF2 ACTIVATORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2020-08-20 WO disclosed