SCHEMBL22367476

SCHEMBL22367476

O=C1NCCN(C(F)(F)F)c2ncccc21

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 12/20 0.43
EPHX2 P34913 1/20 0.41
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
POLB P06746 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
MAPK1 P28482 1/20 0.37
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
PDE3A Q14432 1/20 0.37
PDPK1 O15530 1/20 0.36
PARP10 Q53GL7 1/20 0.36
PARP11 Q9NR21 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22367242 0.77 PARP1 (0.46) PARP1ALDH1A1LMNAPOLBADORA3
SCHEMBL22322734 0.68 ALDH1A1 (0.40) EPHX2ALDH1A1LMNAPOLBADORA3
SCHEMBL26605078 0.65 ALDH1A1 (0.34) ALDH1A1POLB
SCHEMBL699878 0.65 CYP1A2 (0.58) PARP1ALDH1A1PDPK1PARP10PARP11
SCHEMBL26915147 0.65 HTR2C (0.56)
SCHEMBL31244884 0.65 HTR2C (0.56)
SCHEMBL11584126 0.65 EPHX2 (0.41) EPHX2PDE3A
SCHEMBL14192117 0.65 PARP1 (0.42) PARP1PDPK1PARP10PARP11
SCHEMBL11738800 0.64 KMT2A (0.43) ALDH1A1LMNAPOLBADORA3MAPK1
SCHEMBL299004 0.64 PARP1 (0.53) PARP1PDPK1PARP10PARP11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3700890-A1 NEW ALCOXYAMINO DERIVATIVES FOR TREATING PAIN AND PAIN RELATED CONDITIONS ESTEVE PHARMACEUTICALS, S.A. (ES) 2020-09-02 EP claimed
EP-3700890-A1 NEW ALCOXYAMINO DERIVATIVES FOR TREATING PAIN AND PAIN RELATED CONDITIONS ESTEVE PHARMACEUTICALS, S.A. (ES) 2020-09-02 EP disclosed