SCHEMBL22397156

SCHEMBL22397156

CCOC(=O)C1=CNNC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.42
MEN1 O00255 3/20 0.42
KDM4E B2RXH2 3/20 0.42
MAPT P10636 3/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.41
CA12 O43570 3/20 0.39
CA1 P00915 3/20 0.39
CA2 P00918 3/20 0.39
CA7 P43166 3/20 0.39
CA9 Q16790 3/20 0.39
CA14 Q9ULX7 3/20 0.39
ESR1 P03372 1/20 0.39
ESR2 Q92731 1/20 0.39
CYP1A2 P05177 3/20 0.38
LMNA P02545 3/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
NR1H2 P55055 1/20 0.38
NR1H3 Q13133 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16863288 0.75 KMT2A (0.40) KMT2AMEN1KDM4EMAPTALOX15
SCHEMBL1284263 0.75 ALDH1A1 (0.41) KMT2AMEN1KDM4EMAPTALOX15
SCHEMBL9797391 0.73 KDM4E (0.48) KMT2AMEN1KDM4EMAPTALOX15
SCHEMBL20161452 0.73 FUCA1 (0.39) KMT2AMEN1KDM4EMAPTALOX15
SCHEMBL23757667 0.73 ATM (0.42) KMT2AMEN1KDM4EMAPTALOX15
SCHEMBL4448027 0.70 KMT2A (0.42) KMT2AMEN1KDM4EMAPTALOX15
SCHEMBL12659213 0.70 CHRM3 (0.43) KMT2AMEN1KDM4EMAPTALOX15
SCHEMBL10447298 0.70 TSHR (0.48) KMT2AMEN1KDM4EMAPTALOX15
SCHEMBL43932 0.70
SCHEMBL29093155 0.69 KMT2A (0.40) KMT2AMEN1KDM4EMAPTALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3704112-A1 ALKENE SPIROCYCLIC COMPOUNDS AS FARNESOID X RECEPTOR MODULATORS Bristol-Myers Squibb Company (US) 2020-09-09 EP disclosed