SCHEMBL22397178

SCHEMBL22397178

CC(C)(F)Oc1ccc(C#N)nc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.43
AR P10275 1/20 0.38
SLC40A1 Q9NP59 1/20 0.36
CHEK1 O14757 6/20 0.35
DGAT1 O75907 1/20 0.35
ALOX5AP P20292 1/20 0.34
FEN1 P39748 1/20 0.34
NSD2 O96028 1/20 0.34
NSD3 Q9BZ95 1/20 0.34
NQO1 P15559 1/20 0.33
PDE10A Q9Y233 1/20 0.33
SLC22A12 Q96S37 1/20 0.32
CTSS P25774 1/20 0.32
KCNQ3 O43525 1/20 0.32
KCNQ2 O43526 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
HPGD P15428 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL506801 0.86 TRPA1 (0.41) TRPA1ARSLC40A1CHEK1DGAT1
SCHEMBL29620884 0.85 TRPA1 (0.55) TRPA1ARSLC40A1DGAT1ALOX5AP
SCHEMBL11894343 0.85 AR (0.39) TRPA1ARSLC40A1CHEK1ALOX5AP
SCHEMBL10329121 0.85 TRPA1 (0.55) TRPA1ARSLC40A1DGAT1ALOX5AP
SCHEMBL10329120 0.82 TRPA1 (0.43) TRPA1ARSLC40A1CHEK1DGAT1
SCHEMBL19767081 0.79 AR (0.39) TRPA1ARSLC40A1CHEK1DGAT1
SCHEMBL17162369 0.78 AR (0.41) TRPA1ARSLC40A1CHEK1DGAT1
SCHEMBL21174927 0.77 TRPA1 (0.40) TRPA1SLC40A1CHEK1DGAT1ALOX5AP
SCHEMBL29601639 0.75 TRPA1 (0.40) TRPA1ARCHEK1DGAT1NSD2
SCHEMBL17395028 0.75 TRPA1 (0.40) TRPA1ARCHEK1DGAT1NSD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3704112-A1 ALKENE SPIROCYCLIC COMPOUNDS AS FARNESOID X RECEPTOR MODULATORS Bristol-Myers Squibb Company (US) 2020-09-09 EP disclosed