SCHEMBL22397180

SCHEMBL22397180

O=C(O)c1cc(OC2CCOC2)c2ccccc2n1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.56
PDE4D Q08499 11/20 0.44
PDE4A P27815 6/20 0.44
PDE4B Q07343 6/20 0.44
PDE4C Q08493 6/20 0.44
GRM5 P41594 2/20 0.42
MAPK1 P28482 2/20 0.40
KAT2B Q92831 1/20 0.40
BAZ2B Q9UIF8 1/20 0.40
POLB P06746 1/20 0.39
NTRK1 P04629 1/20 0.39
NTRK3 Q16288 1/20 0.39
NTRK2 Q16620 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30421897 1.00 ALOX15 (0.56) ALOX15PDE4DPDE4APDE4BPDE4C
SCHEMBL30421034 1.00 ALOX15 (0.56) ALOX15PDE4DPDE4APDE4BPDE4C
SCHEMBL30421104 0.90 ALOX15 (0.61) ALOX15GRM5POLB
SCHEMBL22392805 0.84 EGFR (0.45) ALOX15PDE4DPDE4APDE4BPDE4C
SCHEMBL22392856 0.84 EGFR (0.45) ALOX15PDE4DPDE4APDE4BPDE4C
SCHEMBL22392807 0.84 EGFR (0.45) ALOX15PDE4DPDE4APDE4BPDE4C
SCHEMBL29469533 0.78 ALOX15 (0.59) ALOX15POLB
SCHEMBL30420987 0.77 ALOX15 (0.58) ALOX15POLB
SCHEMBL1201785 0.76 GRM5 (0.50) GRM5
SCHEMBL6818987 0.75 NPC1 (0.47) ALOX15PDE4DPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3704112-A1 ALKENE SPIROCYCLIC COMPOUNDS AS FARNESOID X RECEPTOR MODULATORS Bristol-Myers Squibb Company (US) 2020-09-09 EP disclosed