SCHEMBL22397202

SCHEMBL22397202

O=C1N[C@@H](O)c2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.51
HTR2A P28223 2/20 0.49
HTR2C P28335 2/20 0.49
HTR2B P41595 2/20 0.49
PARP1 P09874 1/20 0.49
CYP1A2 P05177 1/20 0.45
PARP3 Q9Y6F1 1/20 0.45
TNKS2 Q9H2K2 5/20 0.44
TSHR P16473 2/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
PBRM1 Q86U86 1/20 0.44
IDO1 P14902 1/20 0.41
GSK3B P49841 1/20 0.41
KMT2A Q03164 1/20 0.41
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29941489 1.00 HSD17B10 (0.51) HSD17B10HTR2AHTR2CHTR2BPARP1
SCHEMBL30179824 1.00 HSD17B10 (0.51) HSD17B10HTR2AHTR2CHTR2BPARP1
SCHEMBL4082700 1.00 HSD17B10 (0.51) HSD17B10HTR2AHTR2CHTR2BPARP1
Phenol SCHEMBL29155438 0.91 KMT2A (0.46) HSD17B10HTR2AHTR2CHTR2BPARP1
SCHEMBL16213357 0.79 PARP1 (0.50) HSD17B10HTR2AHTR2CHTR2BPARP1
SCHEMBL22011499 0.78 GSK3B (0.46) HSD17B10HTR2AHTR2CHTR2BPARP1
SCHEMBL8163254 0.75 HSD17B10 (0.61) HSD17B10HTR2AHTR2CHTR2BPARP1
SCHEMBL18215410 0.75 HSD17B10 (0.61) HSD17B10HTR2AHTR2CHTR2BPARP1
SCHEMBL22268104 0.74 HTR2A (0.35) HSD17B10HTR2AHTR2CHTR2BPARP1
SCHEMBL19573960 0.74 TNKS2 (0.49) HSD17B10HTR2AHTR2CHTR2BPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3704091-A1 MODULATORS OF THE INTEGRATED STRESS PATHWAY Calico Life Sciences LLC (US) 2020-09-09 EP disclosed