SCHEMBL22011499

SCHEMBL22011499

O=C1NC(O)C(=O)c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.46
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
S100A4 P26447 1/20 0.43
POLB P06746 1/20 0.43
TNKS2 Q9H2K2 4/20 0.41
MAPT P10636 2/20 0.40
TSHR P16473 2/20 0.40
HTR2B P41595 2/20 0.40
CASP3 P42574 1/20 0.40
CASP2 P42575 1/20 0.40
CASP7 P55210 1/20 0.40
CASP6 P55212 1/20 0.40
CASP8 Q14790 1/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
MAPK1 P28482 1/20 0.40
HSD17B10 Q99714 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31739367 0.80 TSHR (0.47) KMT2AMEN1S100A4POLBTNKS2
SCHEMBL19492450 0.80 TSHR (0.47) KMT2AMEN1S100A4POLBTNKS2
SCHEMBL22397202 0.78 HSD17B10 (0.51) GSK3BKMT2ATNKS2TSHRHTR2B
SCHEMBL4082700 0.78 HSD17B10 (0.51) GSK3BKMT2ATNKS2TSHRHTR2B
SCHEMBL29941489 0.78 HSD17B10 (0.51) GSK3BKMT2ATNKS2TSHRHTR2B
SCHEMBL30179824 0.78 HSD17B10 (0.51) GSK3BKMT2ATNKS2TSHRHTR2B
SCHEMBL8293271 0.74 TSHR (0.48) GSK3BKMT2AMEN1S100A4POLB
SCHEMBL8585951 0.74 MAPT (0.44) GSK3BKMT2AMEN1S100A4POLB
SCHEMBL125094 0.74 MAPT (0.44) GSK3BKMT2AMEN1S100A4POLB
SCHEMBL8090678 0.72 HSD17B10 (0.46) GSK3BKMT2AMEN1S100A4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110028448-B Preparation method of 3-hydroxy-2,3-dihydroisoquinoline-1, 4-diketone compound 嘉兴学院 2020-07-31 CN claimed
CN-110028448-A A kind of preparation method of 3- hydroxyl -2,3- dihydro-isoquinoline -1,4- dione compounds 嘉兴学院 2019-07-19 CN claimed
CN-110028448-B Preparation method of 3-hydroxy-2,3-dihydroisoquinoline-1, 4-diketone compound 嘉兴学院 2020-07-31 CN disclosed
WO-2020102245-A1 IN-FLOW PHOTOOXYGENATION OF AMINOTHIENOPYRIDINONES GENERATES NOVEL PTP4A3 PHOSPHATASE INHIBITORS UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2020-05-22 WO disclosed
WO-2020102243-A2 IN-FLOW PHOTOOXYGENATION OF AMINOTHIENOPYRIDINONES GENERATES NOVEL PTP4A3 PHOSPHATASE INHIBITORS UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2020-05-22 WO disclosed
CN-110028448-A A kind of preparation method of 3- hydroxyl -2,3- dihydro-isoquinoline -1,4- dione compounds 嘉兴学院 2019-07-19 CN disclosed
CN-110028448-A A kind of preparation method of 3- hydroxyl -2,3- dihydro-isoquinoline -1,4- dione compounds 嘉兴学院 2019-07-19 CN disclosed