SCHEMBL22398136

SCHEMBL22398136

OC(CCCn1ccnn1)c1ccc(OCc2coc(C=Cc3ccc(Br)cc3F)n2)cc1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 1/20 0.50
MINK1 Q8N4C8 1/20 0.50
FGFR1 P11362 2/20 0.34
FLT1 P17948 2/20 0.34
FGFR2 P21802 2/20 0.34
FGFR4 P22455 2/20 0.34
FGFR3 P22607 2/20 0.34
FLT4 P35916 2/20 0.34
KDR P35968 2/20 0.34
EGFR P00533 1/20 0.34
PDGFRB P09619 1/20 0.34
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
CYP19A1 P11511 4/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22398133 1.00 ERBB2 (0.50) ERBB2MINK1FGFR1FLT1FGFR2
SCHEMBL26316603 0.91 ERBB2 (0.52) ERBB2MINK1
SCHEMBL22398070 0.90 ERBB2 (0.60) ERBB2MINK1
SCHEMBL28470367 0.90 ERBB2 (0.60) ERBB2MINK1
SCHEMBL22398054 0.88 ERBB2 (0.47) ERBB2MINK1CYP19A1
SCHEMBL28476214 0.88 ERBB2 (0.47) ERBB2MINK1CYP19A1
SCHEMBL26316561 0.87 ERBB2 (0.66) ERBB2MINK1FGFR1FLT1FGFR2
SCHEMBL31130669 0.87 ERBB2 (0.66) ERBB2MINK1FGFR1FLT1FGFR2
SCHEMBL22398061 0.87 ERBB2 (0.66) ERBB2MINK1FGFR1FLT1FGFR2
SCHEMBL28470352 0.86 ERBB2 (0.49) ERBB2MINK1FGFR1FLT1FGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111886234-A Heterocyclic mitochondrial activity inhibitors and uses thereof 蒙特利尔大学 2020-11-03 CN disclosed
EP-3704111-A1 HETEROCYCLIC MITOCHONDRIAL ACTIVITY INHIBITORS AND USES THEREOF Université de Montréal (CA) 2020-09-09 EP disclosed