SCHEMBL28470352

SCHEMBL28470352

O=C(CCCn1ccnn1)c1ccc(OCc2coc(C=Cc3ccc(Br)cc3F)n2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 1/20 0.49
MINK1 Q8N4C8 1/20 0.49
FGFR1 P11362 2/20 0.33
FLT1 P17948 2/20 0.33
FGFR2 P21802 2/20 0.33
FGFR4 P22455 2/20 0.33
FGFR3 P22607 2/20 0.33
FLT4 P35916 2/20 0.33
KDR P35968 2/20 0.33
EGFR P00533 1/20 0.33
PDGFRB P09619 1/20 0.33
PTGS2 P35354 2/20 0.33
ALOX5AP P20292 1/20 0.31
FFAR1 O14842 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
HDAC3 O15379 1/20 0.30
HDAC4 P56524 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC7 Q8WUI4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22398008 1.00 ERBB2 (0.49) ERBB2MINK1FGFR1FLT1FGFR2
SCHEMBL26316601 0.91 ERBB2 (0.51) ERBB2MINK1FFAR1NPC1RAB9A
SCHEMBL28472619 0.90 ERBB2 (0.59) ERBB2MINK1FFAR1
SCHEMBL22397911 0.90 ERBB2 (0.59) ERBB2MINK1FFAR1
SCHEMBL22398048 0.88 ERBB2 (0.47) ERBB2MINK1RAB9A
SCHEMBL22398043 0.88 ERBB2 (0.47) ERBB2MINK1RAB9A
SCHEMBL26316561 0.86 ERBB2 (0.66) ERBB2MINK1FGFR1FLT1FGFR2
SCHEMBL31130669 0.86 ERBB2 (0.66) ERBB2MINK1FGFR1FLT1FGFR2
SCHEMBL22398061 0.86 ERBB2 (0.66) ERBB2MINK1FGFR1FLT1FGFR2
SCHEMBL22398136 0.86 ERBB2 (0.50) ERBB2MINK1FGFR1FLT1FGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111886234-A Heterocyclic mitochondrial activity inhibitors and uses thereof 蒙特利尔大学 2020-11-03 CN disclosed