SCHEMBL2242020

SCHEMBL2242020

Nc1cc([N+](=O)[O-])ccc1S

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.60
TSHR P16473 3/20 0.60
GAA P10253 2/20 0.60
THRB P10828 1/20 0.60
TDP1 Q9NUW8 9/20 0.59
ALDH1A1 P00352 6/20 0.57
ALOX15 P16050 2/20 0.55
HTT P42858 1/20 0.52
MEN1 O00255 3/20 0.49
MAPT P10636 3/20 0.49
KMT2A Q03164 3/20 0.49
GFER P55789 2/20 0.49
LMNA P02545 1/20 0.46
POLB P06746 2/20 0.46
KDM4E B2RXH2 1/20 0.46
ATM Q13315 1/20 0.46
APEX1 P27695 1/20 0.46
CASP6 P55212 1/20 0.46
CTDSP1 Q9GZU7 1/20 0.46
HSD17B10 Q99714 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5973685 0.98 CYP3A4 (0.58) CYP3A4TSHRGAATHRBTDP1
SCHEMBL27543233 0.98 CYP3A4 (0.58) CYP3A4TSHRGAATHRBTDP1
SCHEMBL27518040 0.98 CYP3A4 (0.58) CYP3A4TSHRGAATHRBTDP1
SCHEMBL392484 0.85 TDP1 (0.61) CYP3A4TSHRGAATHRBTDP1
SCHEMBL29353815 0.82 CYP3A4 (0.69) CYP3A4TSHRGAATHRBTDP1
SCHEMBL78293 0.82 CYP3A4 (0.69) CYP3A4TSHRGAATHRBTDP1
Methane SCHEMBL28785435 0.80 CYP3A4 (0.67) CYP3A4TSHRGAATHRBTDP1
Hydrochloric Acid SCHEMBL970605 0.80 CYP3A4 (0.67) CYP3A4TSHRGAATHRBTDP1
SCHEMBL11822059 0.80 TSHR (0.52) CYP3A4TSHRGAATHRBTDP1
SCHEMBL31435677 0.80 CYP3A4 (0.67) CYP3A4TSHRGAATHRBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 65 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113754606-A Phenoxazinediamine derivatives and/or phenothiazine diamine derivatives and preparation method thereof 南京工业大学 2021-12-07 CN claimed
WO-2022213975-A1 COMPOUNDS TARGETING Y220C MUTANT OF P53 JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2022-10-13 WO disclosed
CN-114656418-A (E) -benzo five-membered ring-styryl sulfonium salt derivatives, and preparation and application thereof 同济大学 2022-06-24 CN disclosed
CN-111138380-B Method for continuously synthesizing benzothiadiazole compound 浙江工业大学 2022-02-15 CN disclosed
CN-113754606-A Phenoxazinediamine derivatives and/or phenothiazine diamine derivatives and preparation method thereof 南京工业大学 2021-12-07 CN disclosed
CN-111138380-A Method for continuously synthesizing benzothiadiazole compound 浙江工业大学 2020-05-12 CN disclosed
EP-3251694-A1 DRUG COMBINATIONS FOR THE TREATMENT OF DUCHENNE MUSCULAR DYSTROPHY Summit (Oxford) Limited (GB) 2017-12-06 EP disclosed
US-20170155053-A1 Molecular and Polymeric Semiconductors and Related Devices USINVEST LLC 2017-06-01 US disclosed
WO-2016025632-A1 MOLECULAR AND POLYMERIC SEMICONDUCTORS AND RELATED DEVICES POLYERA CORPORATION (US) 2016-02-18 WO disclosed
EP-1986633-B1 TREATMENT OF DUCHENNE MUSCULAR DYSTROPHY SUMMIT CORP PLC (GB) 2014-07-30 EP disclosed
EP-0116827-B1 PROCESS FOR THE PREPARATION OF BENZOTHIAZOLES BAYER AG (DE) 1991-04-10 EP disclosed
US-4978476-A Side chain polymers exhibiting nonlinear optical response HOECHST CELANESE CORP. (US) 1990-12-18 US disclosed
US-4808723-A Process for the preparation of benzothiazoles BAYER AKTIENGESELLSCHAFT (DE) 1989-02-28 US disclosed
EP-0061082-B1 PROCESS FOR THE PREPARATION OF 2,3-DIHYDRO-4H-1,4-BENZOTHIAZINES BAYER AG (DE) 1984-11-28 EP disclosed
EP-0116827-A2 Process for the preparation of benzothiazoles BAYER AG (DE) 1984-08-29 EP disclosed
US-4393206-A DEHYDROCYCLIZATION OF 2-(2-HYDROXYALKYL)-THIOANILINES BAYER AKTIENGESELLSCHAFT (DE) 1983-07-12 US disclosed
EP-0061082-A1 Process for the preparation of 2,3-dihydro-4H-1,4-benzothiazines BAYER AG (DE) 1982-09-29 EP disclosed
US-4137228-A HIGH TINCTORIAL STRENGTH, COLORFASTNESS CASSELLA AKTIENGESELLSCHAFT (DE) 1979-01-30 US disclosed
US-4033945-A Water-soluble trisazo 8-amino-naphthol-1 dyes CASSELLA FARBWERKE MAINKUR AKTIENGESELLSCHAFT (DT) 1977-07-05 US disclosed
US-3985885-A ANTHELMINTIC AGENTS E. R. SQUIBB & SONS, INC. (US) 1976-10-12 US disclosed