SCHEMBL22426005

SCHEMBL22426005

CC(C)(C)OC(=O)NC1C=C[C@H](N)C1

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 5/20 0.55
NFKB2 Q00653 5/20 0.55
RELA Q04206 5/20 0.55
BTK Q06187 1/20 0.43
KDM1A O60341 2/20 0.40
GAA P10253 1/20 0.39
MAOB P27338 1/20 0.38
EPHX2 P34913 1/20 0.38
CTSK P43235 2/20 0.37
KMT2A Q03164 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23912305 1.00 NFKB1 (0.55) NFKB1NFKB2RELABTKKDM1A
SCHEMBL22084065 1.00 NFKB1 (0.55) NFKB1NFKB2RELABTKKDM1A
SCHEMBL22242697 1.00 NFKB1 (0.55) NFKB1NFKB2RELABTKKDM1A
SCHEMBL4714078 0.85 NFKB1 (0.54) NFKB1NFKB2RELABTKKDM1A
SCHEMBL4714074 0.85 NFKB1 (0.54) NFKB1NFKB2RELABTKKDM1A
SCHEMBL4714079 0.85 NFKB1 (0.54) NFKB1NFKB2RELABTKKDM1A
SCHEMBL22084467 0.83 NFKB1 (0.55) NFKB1NFKB2RELABTKKDM1A
SCHEMBL14586680 0.83 NFKB1 (0.55) NFKB1NFKB2RELABTKKDM1A
SCHEMBL2630497 0.83 NFKB1 (0.55) NFKB1NFKB2RELABTKKDM1A
SCHEMBL22084627 0.83 NFKB1 (0.55) NFKB1NFKB2RELABTKKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11248001-B2 PCSK9 inhibitors and methods of use thereof ASTRAZENECA AB (SE) 2022-02-15 US disclosed
US-20200291041-A1 PCSK9 Inhibitors and Methods of Use Thereof ASTRAZENECA AB (SE) 2020-09-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11248001-B2 PCSK9 inhibitors and methods of use thereof PCSK9, PCSK7, PCSK6 NFKB1 1341/4885NFKB2 1376/4885RELA 934/4885
US-20200291041-A1 PCSK9 Inhibitors and Methods of Use Thereof PCSK9, PCSK7, PCSK6 NFKB1 1500/4885NFKB2 1545/4885RELA 900/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.