SCHEMBL224277

SCHEMBL224277

Fc1cc(Br)ccc1OCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.55
CCR5 P51681 5/20 0.54
SLC6A4 P31645 1/20 0.54
MAOB P27338 1/20 0.53
ALDH1A1 P00352 3/20 0.52
USP28 Q96RU2 1/20 0.52
USP25 Q9UHP3 1/20 0.52
RAB9A P51151 1/20 0.52
HTT P42858 2/20 0.51
LRRK2 Q5S007 1/20 0.51
PTGER1 P34995 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.49
S1PR5 Q9H228 1/20 0.48
LMNA P02545 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30739242 1.00 KDM1A (0.55) KDM1ACCR5SLC6A4MAOBALDH1A1
SCHEMBL8617145 0.89 ERN1 (0.53) KDM1ACCR5SLC6A4MAOBALDH1A1
SCHEMBL8619252 0.89 ERN1 (0.53) KDM1ACCR5SLC6A4MAOBALDH1A1
SCHEMBL8612822 0.89 ERN1 (0.48) KDM1ACCR5SLC6A4MAOBALDH1A1
SCHEMBL8616532 0.89 KDM1A (0.46) KDM1ACCR5SLC6A4MAOBALDH1A1
SCHEMBL8617807 0.89 KDM1A (0.46) KDM1ACCR5SLC6A4MAOBALDH1A1
SCHEMBL8613905 0.86 ERN1 (0.47) KDM1ACCR5SLC6A4MAOBALDH1A1
SCHEMBL29704022 0.86 KDM1A (0.55) KDM1ACCR5SLC6A4MAOBALDH1A1
SCHEMBL15057279 0.86 KDM1A (0.55) KDM1ACCR5SLC6A4MAOBALDH1A1
SCHEMBL8643887 0.85 ERN1 (0.48) KDM1ACCR5SLC6A4MAOBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 185 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250388575-A1 HETEROBIFUNCTIONAL COMPOUNDS AND METHODS OF TREATING DISEASE HALDA THERAPEUTICS OPCO INC (US) 2025-12-25 US disclosed
WO-2024213125-A1 BRM SELECTIVE DEGRADATION AGENT AND USE THEREOF 南京再明医药有限公司 2024-10-17 WO disclosed
WO-2024054955-A1 HETEROBIFUNCTIONAL COMPOUNDS AND METHODS OF TREATING DISEASE HALDA THERAPEUTICS OPCO, INC. (US) 2024-03-14 WO disclosed
WO-2024054955-A1 HETEROBIFUNCTIONAL COMPOUNDS AND METHODS OF TREATING DISEASE HALDA THERAPEUTICS OPCO, INC. (US) 2024-03-14 WO disclosed
CN-117466897-A Highly selective FGFR2 inhibitors 深圳福沃药业有限公司 2024-01-30 CN disclosed
CN-107722996-B Polymerizable liquid crystal compound and preparation method and application thereof 北京八亿时空液晶科技股份有限公司 2023-06-09 CN disclosed
US-11274100-B2 EP300/CREBBP inhibitor DAIICHI SANKYO COMPANY, LIMITED (JP) 2022-03-15 US disclosed
CN-107699252-B Polymeric liquid crystal compound and preparation method and application thereof 北京八亿时空液晶科技股份有限公司 2021-09-07 CN disclosed
US-20210171520-A1 EP300/CREBBP INHIBITOR DAIICHI SANKYO COMPANY, LIMITED (JP) 2021-06-10 US disclosed
US-20210121453-A1 SELECTIVE NR2B ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2021-04-29 US disclosed
WO-1994010179-A1 ARYLBORON ACIDS AS INTERMEDIATES IN THE PRODUCTION OF COMPONENTS OF LIQUID-CRYSTAL MIXTURES HOECHST AKTIENGESELLSCHAFT (DE) 1994-05-11 WO disclosed
US-5182047-A FLUORINATED BIPHENYLDIOLE DERIVATIVES MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 1993-01-26 US disclosed
EP-0368975-B1 FLUORINATED BIPHENYLDIOLE DERIVATIVES MERCK PATENT GmbH (DE) 1992-12-16 EP disclosed
EP-0496896-A1 CYCLOBUTANECARBOXYLIC ACID DERIVATIVE AND LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME KANTO KAGAKU KABUSHIKI KAISHA (JP) 1992-08-05 EP disclosed
EP-0394906-A2 Liquid crystalline composition MERCK PATENT GmbH (DE) 1990-10-31 EP disclosed
EP-0388141-A1 Ferroelectric liquid crystal device SHARP KABUSHIKI KAISHA (JP) 1990-09-19 EP disclosed
EP-0385662-A2 Heterocycles with inhibitory activity of 5-lipoxygenase ZENECA LIMITED (GB) 1990-09-05 EP disclosed
EP-0375404-A2 Heterocyclic derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-06-27 EP disclosed
EP-0368975-A1 FLUORINATED BIPHENYLDIOLE DERIVATIVES. MERCK PATENT GMBH (DE) 1990-05-23 EP disclosed
WO-1989012039-A1 FLUORINATED BIPHENYLDIOLE DERIVATIVES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1989-12-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11274100-B2 EP300/CREBBP inhibitor EP300, CREBBP, CREB1 KDM1A 216/4885CCR5 3243/4885SLC6A4 3517/4885
US-20250388575-A1 HETEROBIFUNCTIONAL COMPOUNDS AND METHODS OF TREATING DISEASE H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, HCCS, CBR1 KDM1A 3155/4885CCR5 56/4885SLC6A4 3204/4885
US-20210121453-A1 SELECTIVE NR2B ANTAGONISTS GRIN2B, GRIN2A, GRIN3A KDM1A 4138/4885CCR5 2377/4885SLC6A4 220/4885
US-20210171520-A1 EP300/CREBBP INHIBITOR EP300, CREBBP, CREB1 KDM1A 216/4885CCR5 3243/4885SLC6A4 3517/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.