SCHEMBL22428786

SCHEMBL22428786

CNc1nc(NC2CCCC2)c2ncccc2n1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GPR39 O43194 2/20 0.48
KDM4E B2RXH2 1/20 0.44
GAA P10253 1/20 0.44
NPY5R Q15761 1/20 0.43
MERTK Q12866 6/20 0.43
AXL P30530 1/20 0.43
TYRO3 Q06418 1/20 0.43
ADORA3 P0DMS8 2/20 0.42
ADORA2A P29274 2/20 0.42
ADORA1 P30542 2/20 0.42
KMT2A Q03164 1/20 0.41
PDE4A P27815 1/20 0.41
TLR7 Q9NYK1 2/20 0.41
MAPK8 P45983 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22411318 0.82 TYRO3 (0.59) MERTKAXLTYRO3TLR7
SCHEMBL22411411 0.81 KMT2A (0.47) KDM4EGAAADORA3ADORA2AADORA1
SCHEMBL22872852 0.80 KMT2A (0.49) KDM4EGAAADORA3ADORA2AADORA1
SCHEMBL22411415 0.78 JAK2 (0.39) KDM4EGAAMERTKADORA3ADORA2A
SCHEMBL22872907 0.78 GBA1 (0.49)
SCHEMBL22411399 0.77 CTSL (0.52)
SCHEMBL22872905 0.75 LATS1 (0.60) KDM4EKMT2A
SCHEMBL22428693 0.75 TLR8 (0.38) MERTKADORA3ADORA2ATLR7MAPK8
SCHEMBL22411416 0.74 MAPK8 (0.38) KDM4EGAAADORA3ADORA2APDE4A
SCHEMBL22872893 0.74 MAP4K4 (0.49) KDM4EGAAADORA3ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020185738-A1 HETEROAROMATIC AND HETEROBICYCLIC AROMATIC DERIVATIVES FOR THE TREATMENT OF FERROPTOSIS-RELATED DISORDERS COLLABORATIVE MEDICINAL DEVELOPMENT, LLC (US) 2020-09-17 WO disclosed