SCHEMBL22447486

SCHEMBL22447486

COC(=O)C(F)(F)Cn1cnc2ccc(Br)cc2c1=O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.56
LMNA P02545 1/20 0.53
DDR1 Q08345 2/20 0.46
PIK3CA P42336 1/20 0.44
RAB9A P51151 1/20 0.41
MMP13 P45452 2/20 0.41
HDAC6 Q9UBN7 3/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
TSHR P16473 1/20 0.40
HTT P42858 1/20 0.40
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22447490 0.87 MCL1 (0.60) MCL1LMNADDR1RAB9AMMP13
SCHEMBL22447483 0.85 MCL1 (0.54) MCL1LMNADDR1PIK3CARAB9A
SCHEMBL31723379 0.80 MCL1 (0.56) MCL1LMNADDR1RAB9AHDAC6
SCHEMBL30987319 0.79 MCL1 (0.58) MCL1LMNADDR1RAB9AHTT
SCHEMBL12933340 0.79 MCL1 (0.57) MCL1LMNADDR1RAB9AHTT
SCHEMBL22447583 0.78 MCL1 (0.57) MCL1LMNADDR1PIK3CARAB9A
SCHEMBL4210572 0.77 MCL1 (0.61) MCL1LMNADDR1RAB9AHTT
SCHEMBL13820349 0.77 MCL1 (0.56) MCL1LMNADDR1RAB9ATNF
SCHEMBL22447510 0.76 MCL1 (0.60) MCL1LMNADDR1RAB9AMMP13
SCHEMBL22447414 0.76 MCL1 (0.64) MCL1LMNAPIK3CARAB9AMMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3712143-A1 QUINAZOLINONE COMPOUND AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2020-09-23 EP disclosed