SCHEMBL22450554

SCHEMBL22450554

CC1CCN(C(=O)c2cnc3c(c2)nc(-c2cc4cccnc4n2CC2CC2)n3C)CC1

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PADI4 Q9UM07 19/20 0.54
PDE4A P27815 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4C Q08493 1/20 0.44
PDE4D Q08499 1/20 0.44
CYP1A2 P05177 1/20 0.44
TSHR P16473 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18975348 0.92 PADI4 (0.59) PADI4
SCHEMBL18975351 0.90 PADI4 (0.56) PADI4PDE4APDE4BPDE4CPDE4D
SCHEMBL18938868 0.88 PADI4 (0.54) PADI4
SCHEMBL22450519 0.86 PADI4 (0.61) PADI4
SCHEMBL18960699 0.86 PADI4 (0.74) PADI4
SCHEMBL22450628 0.86 PADI4 (0.52) PADI4PDE4APDE4BPDE4CPDE4D
SCHEMBL18955611 0.86 PADI4 (0.59) PADI4PDE4APDE4BPDE4CPDE4D
SCHEMBL18960751 0.86 PADI4 (0.59) PADI4PDE4APDE4BPDE4CPDE4D
SCHEMBL18955572 0.86 PADI4 (0.59) PADI4PDE4APDE4BPDE4CPDE4D
SCHEMBL18955613 0.86 PADI4 (0.59) PADI4PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3386505-B1 AZA-BENZIMIDAZOLE INHIBITORS OF PAD4 PADLOCK THERAPEUTICS INC (US) 2020-09-23 EP disclosed